专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

21. 发明授权

US07241721B2 Biphenyl derivatives and their use as fungicides 失效
公开(公告)号：US07241721B2
公开(公告)日：2007-07-10
申请号：US10540036
申请日：2003-12-15
申请人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
IPC分类号： A01N43/56 , C07D231/18
CPC分类号： C07D213/82 , A01N43/06 , A01N43/14 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/74 , A01N43/80 , C07C25/24 , C07C211/45 , C07C211/52 , C07C217/76 , C07C219/32 , C07C233/03 , C07C2601/02 , C07C2601/08 , C07D207/34 , C07D231/14 , C07D231/16 , C07D237/24 , C07D239/28 , C07D239/30 , C07D263/34 , C07D277/56 , C07D307/68 , C07D309/28 , C07D327/06 , C07D333/38 , C07F7/0812
摘要： A fungicidally active compound of formula (I): where Het is a substituted 5- or 6-membered heterocyclic ring; R1 is hydrogen, formyl, CO—C1-4 alkyl, COO—C1-4 alkyl, C1-4 alkoxy(C1-4)alkylene, CO—C1-4 alkylenoxy(C1-4)alkyl, propargyl or allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, methyl or CF3; each R6 is, independently, halogen, methyl or CF3; R7 is (Z)mC═C(Y1), (Z)mC(Y1)═C(Y2)(Y3) or tri(C1-4)alkylsilyl; X is O or S; Y1, Y2 and Y3 are each, independently, hydrogen, halogen, C1-6 alkyl [optionally substituted by one or more substituents each independently selected from halogen, hydroxy, C1-4 alkoxy, C1-4 haloalkoxy, C1-4 alkylthio, C1-4 haloalkylthio, C1-4 alkylamino, di(C1-4)alkylamino, C1-4 alkoxycarbonyl, C1-4 alkylcarbonyloxy and tri(C1-4)alkylsilyl], C2-4 alkenyl [optionally substituted by one or more substituents each independently selected from halogen], C2-4 alkynyl [optionally substituted by one or more substituents each independently selected from halogen], C3-7 cycloalkyl [optionally substituted by one or more substituents each independently selected from halogen, C1-4 alkyl and C1-4 haloalkyl] or tri(C1-4)alkylsilyl; Z is C1-4 alkylene [optionally substituted by one or more substituents each independently selected from hydroxy, cyano, C1-4 alkoxy, halogen, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylthio, COOH and COO—C1-4 alkyl]; m is 0 or 1; and n is 0, 1 or 2; the invention also relates to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi

22. 发明申请

US20060154967A1 Chemical compounds 失效
公开(公告)号：US20060154967A1
公开(公告)日：2006-07-13
申请号：US10524721
申请日：2003-08-18
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/64 , A01N43/40 , C07D417/02 , C07D409/02 , C07D405/02 , C07D403/02
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (I):, where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4 alkyl) (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl (where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4)alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).

23. 发明申请

US20100227898A1 NOVEL MICROBIOCIDES 有权
标题翻译：新型微生物
公开(公告)号：US20100227898A1
公开(公告)日：2010-09-09
申请号：US12665349
申请日：2008-06-30
申请人： Harald Walter , Daniel Stierli , Hans Tobler
发明人： Harald Walter , Daniel Stierli , Hans Tobler
IPC分类号： A01N43/40 , C07D231/18 , A01N43/56 , C07D409/06 , C07D233/64 , A01N43/50 , C07D333/52 , A01N43/12 , A01P1/00
CPC分类号： C07D333/28 , C07D333/62 , C07D409/12 , C07D417/12
摘要： Compounds of the formula (I) in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物适合用作杀微生物剂。

24. 发明申请

US20100222389A1 NOVEL MICROBIOCIDES 失效
标题翻译：新型微生物
公开(公告)号：US20100222389A1
公开(公告)日：2010-09-02
申请号：US12664415
申请日：2008-06-13
申请人： Harald Walter , Daniel Stierli , Hans Tobler
发明人： Harald Walter , Daniel Stierli , Hans Tobler
IPC分类号： A01N43/40 , C07D409/12 , A01N43/56 , A01N43/36 , A01N43/647 , C07D417/12 , A01N43/78 , C07D333/24 , A01N43/10 , C07D333/60 , A01N43/12 , A01P3/00
CPC分类号： C07D333/28 , A01N43/10 , A01N43/12 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/78 , C07D333/62 , C07D409/12 , C07D417/12
摘要： Compounds of the formula (I), in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物适合用作杀微生物剂。

25. 发明申请

US20100204287A1 HETEROCYCLIC AMIDE DERIVATIVES USEFUL AS MICROBIOCIDES 有权
标题翻译：杂环酰胺衍生物作为微生物有用
公开(公告)号：US20100204287A1
公开(公告)日：2010-08-12
申请号：US12765942
申请日：2010-04-23
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
IPC分类号： A01N43/78 , A01P17/00
CPC分类号： C07C205/06 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/76 , A01N43/78 , C07C205/11 , C07C205/12 , C07C205/37 , C07C205/45 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D207/46 , C07D213/89 , C07D231/14 , C07D249/04 , C07D263/34 , C07D277/56 , C07D327/06
摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R6, R7 and R8; R1 is hydrogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, C1-4 haloalkoxy, CH2C≡CR9, CH2CR10═CHR11, CH═C═CH2 or COR12; R2 and R3 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl or C1-4 haloalkoxy; R4 and R5 are each independently selected from halo, cyano and nitro; or one of R4 and R5 is hydrogen and the other is selected from halo, cyano and nitro; R6, R7 and R8 are each, independently, hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 haloalkoxy(C1-4)alkyl or C1-4 haloalkoxy, provided that at least one of R6, R7 and R8 is not hydrogen; R9, R10 and R11 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 alkoxy(C1-4)alkyl; and R12 is hydrogen, C1-6 alkyl, C1-6 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 alkylthio(C1-4)-alkyl, C1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被R6基团取代，R7和R8; R 1是氢，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基，CH 2C≡CR9，CH 2 CR 10 = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地是氢，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R4和R5各自独立地选自卤素，氰基和硝基; 或者R4和R5之一是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4卤代烷氧基（C 1-4）烷基或 C 1-4卤代烷氧基，条件是R 6，R 7和R 8中的至少一个不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4烷氧基（C 1-4）烷基; 和R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4烷硫基（C 1-4） - 烷基，C 1-4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

26. 发明申请

US20090221855A1 PROCESS FOR THE PRODUCTION OF ANILINES 有权
标题翻译：生产过程的过程
公开(公告)号：US20090221855A1
公开(公告)日：2009-09-03
申请号：US12065304
申请日：2006-08-28
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
IPC分类号： C07C211/45
CPC分类号： C07C209/10 , C07C209/62 , C07C2601/02 , C07C211/45 , C07C211/48
摘要： The present invention relates to a process for the preparation of compounds of formula wherein R1, R2 and R3 are each independently of the others hydrogen or C1-C4alkyl, by a) reacting compounds of formula (II) wherein R1, R2 and R3 are as defined for formula (I) and X is bromine or chlorine, with a compound of formula (III) wherein R4 is hydrogen or C1-C4alkyl, in the presence of a base and catalytic amounts of at least one palladium complex compound, to form compounds of formula (IV) wherein R1, R2, R3 and R4 are as defined for formula (I), and b) converting those compounds, using a reducing agent, into compounds of formula (I).
摘要翻译：本发明涉及制备下式化合物的方法，其中R 1，R 2和R 3各自独立地为氢或C 1 -C 4烷基，通过a）使式（Ⅱ）化合物（其中R 1，R 2和R 3为与式（Ⅲ）化合物（其中R 4是氢或C 1 -C 4烷基）在碱和催化量的至少一种钯络合物的存在下形成化合物（I），X是溴或氯，其中R 1，R 2，R 3和R 4如式（I）所定义，并且b）使用还原剂将这些化合物转化为式（I）化合物。

27. 发明授权

US07514584B2 Process for the production of 2(2-aminophenyl)-bicylopropane derivatives 有权
标题翻译：制备2（2-氨基苯基） - 环丙烷衍生物的方法
公开(公告)号：US07514584B2
公开(公告)日：2009-04-07
申请号：US11815895
申请日：2006-02-20
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hermann Schneider , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hermann Schneider , Hans Tobler
IPC分类号： C07C211/00 , C07C205/00
CPC分类号： C07C209/36 , C07C201/12 , C07C303/28 , C07C309/66 , C07C309/67 , C07C2601/02 , C07C211/45 , C07C205/06 , C07C205/11
摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein the substituents are as defined in claim 1, by a) reaction of a compound of formula (II) to form a compound of formula (III) b) reaction of that compound in the presence of a base to form a compound of formula (IV) c) conversion of that compound in the presence of a reducing agent into a compound of formula (I).
摘要翻译：本发明涉及制备式（I）化合物的方法，其中取代基如权利要求1所定义，通过a）式（II）化合物与式（III）化合物的反应b）该化合物在碱存在下反应形成式（Ⅳ）化合物，c）将化合物在还原剂存在下转化成式（I）化合物。

28. 发明申请

US20090069572A1 PROCESS FOR THE PREPARATION OF PYRAZOLES 有权
标题翻译：制备吡唑的方法
公开(公告)号：US20090069572A1
公开(公告)日：2009-03-12
申请号：US11577511
申请日：2005-10-19
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： C07D231/14
CPC分类号： C07D231/14
摘要： The present invention relates to a process for the preparation of compounds of formula I wherein R1 is C1-C4haloalkyl; R2 is C1-C6alkyl and R3 is methyl or ethyl, by reaction of compounds of formula II wherein the substituents are as defined for formula I, with compounds of formula III wherein R3 is as defined for formula I and n is 0 or 1.
摘要翻译：本发明涉及制备式Ⅰ化合物的方法，其中R 1是C 1 -C 4卤代烷基; R 2是C 1 -C 6烷基，R 3是甲基或乙基，其中取代基如式I所定义的式II化合物与式III化合物反应，其中R 3如式I所定义，n是0或1。

29. 发明申请

US20090030233A1 PROCESS FOR THE PRODUCTION OF BIPHENYLS 审中-公开
标题翻译：生产BIPHENYLS的工艺
公开(公告)号：US20090030233A1
公开(公告)日：2009-01-29
申请号：US12092324
申请日：2006-11-13
申请人： Josef Ehrenfreund , Harald Walter , Hans Tobler , Camilla Corsi
发明人： Josef Ehrenfreund , Harald Walter , Hans Tobler , Camilla Corsi
IPC分类号： C07C211/45 , C07C205/06
CPC分类号： C07C201/12 , C07C2601/02 , C07C205/06 , C07C205/11 , C07C205/19 , C07C205/34 , C07C205/42 , C07C205/56
摘要： The present invention relates to a novel process for the preparation of a compound of formula (I): which comprises reacting a compound of formula (II): with a compound of general formula (III): wherein R1 and R2 are H or C1-4 alkyl or R1 and R2 join together to form a C2-3 alkylene group, which is optionally substituted by from 1 to 4 methyl or ethyl groups, or an anhydride of the compound (III), in the presence of a base and of a palladium catalyst which is (a) a palladium (0)- or palladium (II)-triarylphosphine complex optionally in the presence of additional amounts of a triarylphoshine ligand, or (b) a palladium (II) salt in the presence of a triarylphosphine ligand, or (c) metallic palladium, optionally deposited on a support, in the presence of triarylphosphine; there being used from 0.9 to 2 moles of compound (III) for each mole of compound (II).
摘要翻译：本发明涉及制备式（I）化合物的新方法：其包括使式（II）化合物与通式（III）的化合物反应：其中R1和R2是H或C1- 4烷基或R 1和R 2连接在一起形成C2-3亚烷基，其任选被1至4个甲基或乙基取代，或化合物（III）的酸酐，在碱存在下，钯催化剂，其是（a）钯（0） - 或钯（II） - 三芳基膦配合物，任选在另外量的三芳基膦酸配体存在下，或（b）钯（II）盐，在三芳基膦配体，或（c）金属钯，任选地沉积在载体上，在三芳基膦存在下; 对于每摩尔化合物（II），使用0.9至2摩尔的化合物（III）。

30. 发明申请

US20080188442A1 Pyrazole-4-Carboxamide Derivatives as Microbiocides 失效
标题翻译：吡唑-4-甲酰胺衍生物作为杀微生物剂
公开(公告)号：US20080188442A1
公开(公告)日：2008-08-07
申请号：US11996094
申请日：2006-07-17
申请人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/56 , A01N55/10 , C07F7/02 , A01P3/00 , C07D231/06
CPC分类号： C07D409/12 , C07D231/06 , C07D401/12
摘要： Compounds of the formula I in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式I化合物适合用作杀微生物剂。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式