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11. 发明申请

WO2006079556A2 SUBSTITUTED 5-PHENYL PYRIMIDINES I IN THERAPY 审中-公开
标题翻译：取代的5-苯基吡啶在治疗中
公开(公告)号：WO2006079556A2
公开(公告)日：2006-08-03
申请号：PCT/EP2006000774
申请日：2006-01-30
申请人： BASF AG , RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , NAVE BARBARA , SCHIEWECK FRANK , SCHWOEGLER ANJA , JABS THORSTEN , BLETTNER CARSTEN
发明人： RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , NAVE BARBARA , SCHIEWECK FRANK , SCHWOEGLER ANJA , JABS THORSTEN , BLETTNER CARSTEN
IPC分类号： A61K31/506 , A61K31/505 , C07D239/42 , C07D239/48 , C07D401/04 , C07D403/04 , C07D417/04
CPC分类号： C07D239/48 , C07D239/42 , C07D401/04 , C07D403/04 , C07D417/04
摘要： The present invention relates to substituted 5-phenyl pyrimidines I, which carry a radical X in the 4-position of the pyrimidine ring, a radical Y in the 6-position of the pyrimidine ring, the radical X denoting a group of the formula NR 1 R 2 , OR 1a or SR 1a , in which R 1 , R 2 , independently of each other, denote hydrogen, C 1 -C 10 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 10 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -halocycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which radicals may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 ; or the radical NR 1 R 2 may also form a 5- or 6-membered optionally substituted heterocyclic ring, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which are non-adjacent to the nitrogen of NR 1 R 2 , in which two adjacent C atoms or one N atom and one adjacent C atom can be linked by a C 1 -C 4 -alkylene chain and wherein the heterocyclic ring may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 as defined in claim 1, R 1a has one of the meanings given for R 1 except for hydrogen; the radical Y being selected from the group consisting of halogen, cyano, C 1 -C 4 -alkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 4 -alkoxy, C 3 -C 4 -alkenyloxy, C 3 -C 4 -alkynyloxy, C 1 -C 6 -alkylthio, di-(C 1 -C 6 -alkyl)amino or C 1 -C 6 -alkylamino, where the alkyl, alkenyl and alkynyl radicals of Y may be substituted by halogen, cyano, nitro, C 1 -C 2 -alkoxy or C 1 -C 4 -alkoxycarbonyl; and wherein the pyrimidine radical may also carry a radical different from hydrogen in the 2-position and wherein the phenyl ring in the 5-position of the pyrimidine ring may be unsubstituted or carry 1, 2, 3, 4 or 5 radicals L which are different from hydrogen, and the pharmaceutically acceptable salts substituted 5-phenyl pyrimidines for use in therapy, in particular in therapy or treatment of cancerous diseases.
摘要翻译：本发明涉及取代的5-苯基嘧啶I，其在嘧啶环的4-位上携带基团X，嘧啶环的6-位的基团Y，基团X表示式NR的基团其中R 1，R 2，R 2，R 1，R 2， R 2彼此独立地表示氢，C 1 -C 10 - 烷基，C 2 - C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 10 - C 1 -C 3烷基，C 3 -C 8 - 环烷基，C 3 -C 8 - 卤代烷基，C 3 -C 8 - 苯基或含有1,2,3或4个氮原子或1,2或3个氮原子和一个硫或氧原子作为环成员的5-或6-元杂芳基或5-或6-元杂环基，该基团可以未被取代或可以携带1,2,3或4个基团R a1a; 或自由基NR 1 R 2还可以形成含有1,2,3或4个氮原子或1,2或2个氮原子的5或6元任选取代的杂环或3个氮原子和一个硫或氧原子作为环成员，其与NR 1 R 2 O 2的氮不相邻，其中两个相邻的C原子或一个 N原子和一个相邻的C原子可以通过C 1 -C 4 - 亚烷基链连接，并且其中杂环可以是未取代的或可以携带1,2,3 或如权利要求1所定义的4个基团R a1，其中R 1a除了氢之外具有R 1给出的含义之一; 基团Y选自卤素，氰基，C 1 -C 4 - 亚烷基，C 2 -C 3 - 烷基， 4 - 烯基，C 2 -C 4 - 炔基，C 3 -C 6 - 环烷基，C 1 -C 4 - 烷氧基，C 3 -C 4 - 炔基氧基，C 1 -C 4 - 3-C 4 - 炔基氧基，C 1 -C 6 - 烷硫基，二 - （C 1 -C 6） C 1 -C 6 - 烷基）氨基或C 1 -C 6 - 烷基氨基，其中Y的烷基，烯基和炔基可以被卤素，氰基，硝基取代，C 1 -C 2 - 烷氧基或C 1 -C 4 - - 烷氧基; 并且其中嘧啶基团还可以携带2-位上与氢不同的基团，其中嘧啶环的5-位上的苯环可以是未取代的或携带1,2,3,4或5个基团L，其为不同于氢，以及用于治疗，特别是治疗或治疗癌性疾病的药学上可接受的盐取代的5-苯基嘧啶。

12. 发明申请

WO2011117783A3 COMPOSITION FOR PRODUCING MAGNETIC OR MAGNETIZABLE MOLDINGS, AND PROCESS FOR PRODUCING THE SAME 审中-公开
标题翻译：用于生产磁性或可磁性模具的组合物及其制造方法
公开(公告)号：WO2011117783A3
公开(公告)日：2012-07-26
申请号：PCT/IB2011051112
申请日：2011-03-17
申请人： BASF SE , BASF CHINA CO LTD , BLETTNER CARSTEN , KACZUN JUERGEN , KRESS RIA , WIEBELHAUS DAG
发明人： BLETTNER CARSTEN , KACZUN JUERGEN , KRESS RIA , WIEBELHAUS DAG
IPC分类号： H01F1/047 , B22F1/00
CPC分类号： H01F41/0266 , B29C43/003 , H01F1/0558 , H01F1/0578 , H01F1/26 , H01F41/0246
摘要： A composition for producing magnetic or magnetizable moldings, comprising from 95.5 to 98.95% by weight of a powder made of a magnetic or magnetizable material, from 1.0 to 4% by weight of a mixture made of at least one epoxy-novolak resin, and also of at least one hardener, and comprising from 0.05 to 0.5% by weight of at least one additive, based in each case on the total weight of the composition. The mixture made of the at least one epoxy-novolak resin and of the at least one hardener comprises from 85 to 95% by weight of the epoxy-novolak resin and from 5 to 15% by weight of hardener. The hardener has been selected from (cyclo)aliphatic amines and their adducts, polyamides, Mannich bases, amidoamines, phenolic resins, imidazoles, and imidazole derivatives, dicyandiamide, and BF3-monoethanolamine. It also involves a process for producing said composition and a molding made of said composition.
摘要翻译：一种用于生产磁性或可磁化模制品的组合物，其包含95.5至98.95重量％的由磁性或可磁化材料制成的粉末，1.0至4重量％的由至少一种环氧酚醛清漆树脂制成的混合物，以及的至少一种硬化剂，并且包含0.05至0.5重量％的至少一种添加剂，基于每种情况，基于组合物的总重量。由至少一种环氧酚醛清漆树脂和至少一种固化剂制成的混合物包含85-95重量％的环氧酚醛树脂和5-15重量％的硬化剂。固化剂选自（环）脂族胺及其加合物，聚酰胺，曼尼希碱，酰氨基胺，酚醛树脂，咪唑和咪唑衍生物，双氰胺和BF 3 - 单乙醇胺。它还涉及制备所述组合物的方法和由所述组合物制成的模制品。

13. 发明专利

MX287218B Pyrazolecarboxanilides, processes for their preparation and compositions comprising them for controlling harmful fungi 未知
公开(公告)号：MX287218B
公开(公告)日：2011-06-06
申请号：MX7007000854
申请日：2007-07-26
申请人： BASF AG
发明人： BLETTNER CARSTEN , MULLER BERND , HUNGER UDO , GRAMMENOS WASSILIOS , GROTE THOMAS , SCHIEWECK FRANK , STIERL REINHARD , SCHAFER PETER , STRATHMANN SIEGFRIED , RHEINHEIMER JOACHIM , SCHWOGLER ANJA , GEWEHR MARKUS , LOHMANN JAN KLAAS , DIETZ JOCHEN
摘要： The present invention relates to pyrazolecarboxanilides I in which the variables are as defined below: n is zero or 2; m is 2 or 3; X1 is fluorine or chlorine; X2 is halogen; Y is CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p is zero or 1; R1 is fluorine, chlorine, bromine, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen or halogen; R3 is hydrogen, methyl or ethyl; W is O or S; with the proviso that, if a) W=O, R1=methyl and R3 is hydrogen, R2 is not fluorine, or b) W=O, n=0, m=2, p=0, R2 and R3 are hydrogen, R1 is not trifluoromethyl or difluoromethyl, to processes for preparing these compounds, to compositions comprising them and to methods for using them for controlling harmful fungi.

14. 发明专利

ZA200702822B 6-phenyl-7-amino-triazolopyrimidines, methods for the production thereof, the use thereof for controlling pathogenic fungi, and agents containing the same 未知
公开(公告)号：ZA200702822B
公开(公告)日：2009-12-30
申请号：ZA200702822
申请日：2007-04-04
申请人： BASF AG
发明人： BLETTNER CARSTEN , TORMO I BLASCO , JORDI MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , SPEAKMAN JOHN-BRYAN , JABS THORSTEN , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , SCHERER MARIA , STIERL REINHARD , DIETZ JOCHEN
IPC分类号： A01N20100101 , C07D20100101
摘要： 6-Phenyl-7-aminotriazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, which comprises one to four heteroatoms from the group consisting of O, N and S, R 2 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which comprises one to four heteroatoms from the group consisting of O, N and S, R 3 ,R 4 ,R 5 ,R 6 ,R 7 are hydrogen or one of the groups mentioned under R 2 , R 4 , together with R 3 or R 6 , may also form a five- or six-membered saturated or unsaturated ring which, in addition to carbon atoms, may comprise one to three further heteroatoms from the group consisting of O, N and S as ring members; R 2 with R 3 , R 4 with R 5 , R 6 with R 7 may in each case together, with formation of spiro groups, also form a C 2 -C 5 -alkylene, or alkenylene or alkynylene chain which may be interrupted by one to three heteroatoms from the group consisting of O, N and S; p is zero or 1; L is halogen, alkyl, haloalkyl, alkoxy, cyano, nitro, amino, alkylamino, dialkylamino, alkylcarbonylamino, C(O)-R, S(O) n -R; where n is zero, 1 or 2; R is hydrogen, alkyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, amino, alkylamino, dialkylamino; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, alkoxy, alkenyloxy, alkynyloxy or haloalkoxy; Y is oxygen or sulfur; Z is hydrogen, alkyl, haloalkyl, cycloalkyl, alkylcarbonyl, cycloalkylcarbonyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, phenyl, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which comprises one to four heteroatoms from the group consisting of O, N and S; or Z together with R 4 or R 6 may also form a five- or six-membered saturated or unsaturated ring which, in addition to carbon atoms and Y, may comprise one or two further heteroatoms from the group consisting of O, N and S as ring members the groups R 1 to R 7 , Z and R may be substituted according to the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

15. 发明专利

UA87895C2 未知
公开(公告)号：UA87895C2
公开(公告)日：2009-08-25
申请号：UAA200709766
申请日：2006-01-30
申请人： BASF AG
发明人： RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , NAVE BARBARA , SCHIEWECK FRANK , SCHWOEGLER ANJA , JABS THORSTEN , BLETTNER CARSTEN
IPC分类号： A61K31/506 , A61K31/505 , C07D239/42 , C07D239/48 , C07D401/04 , C07D403/04 , C07D417/04

16. 发明专利

EA011360B1 5,6-ДИАЛКИЛ-7-АМИНОТРИАЗОЛОПИРИМИДИНЫ, СПОСОБ ИХ ПОЛУЧЕНИЯ И ИХ ПРИМЕНЕНИЕ ДЛЯ БОРЬБЫ С ПАТОГЕННЫМИ ГРИБАМИ, А ТАКЖЕ СОДЕРЖАЩИЕ ИХ СРЕДСТВА 未知
公开(公告)号：EA011360B1
公开(公告)日：2009-02-27
申请号：EA200601569
申请日：2005-03-08
申请人： BASF AG
发明人： TORMO I BLASCO JORDI , BLETTNER CARSTEN , MULLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHAFER PETER , SCHIEWECK FRANK , SCHWOGLER ANJA , WAGNER OLIVER , NIEDENBRUCK MATTHIAS , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOFL ULRICH , STIERL REINHARD , HUNGER UDO
IPC分类号： C07D487/04
摘要： 5,6-Диалкил-7-аминотриазолопиримидиныформулы Iвкоторойзаместителиимеютследующеезначение: Rозначаеталкил, алкоксиалкил, алкенилилиалкинил; Rозначаеталкил, алкоксилкил, алкенилилиалкинил; причем Rи/или Rзамещенысогласноописанию; способполученияэтихсоединенийи ихприменениедляборьбыс фитопатогеннымигрибами, атакжесредства, содержащиеэтисоединения.

17. 发明专利

NZ547363A 6-(Aminocarbonyl-phenyl) triazolopyrimidines, methods for the production thereof, use thereof for controlling harmful fungi, and substances containing the same 未知
公开(公告)号：NZ547363A
公开(公告)日：2009-01-31
申请号：NZ54736304
申请日：2004-12-17
申请人： BASF AG
发明人： TORMO I BLASCO JORDI , BLETTNER CARSTEN , MULLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHAFER PETER , SCHIEWECK FRANK , SCHWOGLER ANJA , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOFL ULRICH , STIERL REINHARD
IPC分类号： A01N43/90 , C07D487/04
摘要： Disclosed are triazolopyrimidines of formula (I), wherein the substituents have the following meaning: R1, R2 represent hydrogen, alkyl, alkyl halide, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl, or phenyl, naphthyl, or a five-membered to six-membered saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group comprising O, N, and S. R1 and R2 can also form a five-membered or six-membered heterocyclyl or heteroaryl along with the nitrogen atom to which the same are bonded, said heterocyclyl or heteroaryl being bonded via N, while optionally containing an additional heteroatom from the group comprising O, N, and S as a ring member and being optionally substituted according to the description; L represents halogen, cyano, alkyl, alkyl halide, alkoxy, alkenyloxy, or alkoxy carbonyl; m represents 1, 2, 3, or 4, the groups L being optionally different if m is greater than 1; X represents halogen, cyano, alkyl, alkyl halide, alkoxy, or haloalkoxy. Also disclosed are methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant-pathogenic fungi.

18. 发明专利

EA010411B1 5,6-ДИАЛКИЛ-7-АМИНОТРИАЗОЛОПИРИМИДИНЫ, СПОСОБ ИХ ПОЛУЧЕНИЯ И ИХ ПРИМЕНЕНИЕ ДЛЯ БОРЬБЫ С ПАТОГЕННЫМИ ГРИБАМИ, А ТАКЖЕ СОДЕРЖАЩИЕ ИХ СРЕДСТВА 未知
公开(公告)号：EA010411B1
公开(公告)日：2008-08-29
申请号：EA200601619
申请日：2005-03-08
申请人： BASF AG
发明人： TORMO I BLANCO JORDI , BLETTNER CARSTEN , MULLER BERND , GEWEHR MARCUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEIHEIMER JOACHIM , SCHAFER PETER , SCHIEWECK FRANK , SCHWOGLER ANJA , WAGNER OLIVER , NIEDENBRUCK MATTHIAS , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOFL ULRICH , STIERL REINHARD
IPC分类号： C07D487/04 , A01N43/90 , A01P21/00
摘要： 5,6-Диалкил-7-аминотриазолопиримидиныформулы Iвкоторойзаместителиимеютследующеезначение: R- алкилилиалкоксиалкил, причемалифатическиегруппымогутбытьзамещенысогласноописанию; R- CHRCH, циклопропил, СН=СНилиСНСН=СН; R- водород, СНилиСНСН; способполученияэтихсоединений, содержащиеихсредства, атакжеихприменениедляборьбыс фитопатогеннымигрибами.

19. 发明专利

BRPI0516140A 未知
公开(公告)号：BRPI0516140A
公开(公告)日：2008-08-26
申请号：BRPI0516140
申请日：2005-09-27
申请人： BASF AG
发明人： BLETTNER CARSTEN , BLASCO JORDI TORMO L , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , SPEAKMAN JOHN-BRYAN , JABS THORSTEN , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , SCHERER MARIA , STIERL REINHARD , SCHWOEGLER ANJA
IPC分类号： C07D487/04 , A01N43/90

20. 发明专利

NZ545103A 2-Substituted pyrimidines 未知
公开(公告)号：NZ545103A
公开(公告)日：2008-06-30
申请号：NZ54510304
申请日：2004-07-15
申请人： BASF AG
发明人： SCHWOGLER ANJA , GEWEHR MARKUS , MULLER BERND , GROTE THOMAS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , GYPSER ANDREAS , RHEINHEIMER JOACHIM , BLETTNER CARSTEN , SCHAFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , STIERL REINHARD , SCHOFL ULRICH , STRATHMANN SIEGFRIED , SCHERER MARIA
IPC分类号： C07D239/42 , A01N43/54
摘要： Disclosed are compounds of formulae I and V, wherein R4 corresponds to one of formulae (a) and (b) and the remaining substituents are as defined in the specification. Also disclosed is a process for preparing certain compounds of formula I, using compounds of formula V. The compounds I and V are pesticides useful in controlling phytopathogenic fungi.

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