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121. 发明专利

CO5650198A2 TRIAZOLOPIRIMIDINAS 未知
公开(公告)号：CO5650198A2
公开(公告)日：2006-06-30
申请号：CO05128694
申请日：2005-12-21
申请人： BAYER CROPSCIENCE AG
发明人： GEBAUER OLAF , HEINEMANN ULRICH , GREUL JORG NICO , HERRMANN STEFAN , HARTMANN BENOIT , ELBE HANS-LUDWIG , GAYER HERBERT , HILLEBRAND STEFAN , WACHENDORFF NEUMANN ULRIKE , KUCK KARL HEINZ , DAHMEN PETER
IPC分类号： A01N43/90 , A61K31/4196 , A61K31/437 , A61K31/44 , A61K31/505 , C07D213/55 , C07D239/30 , C07D487/04
摘要： 1.- Triazolopirimidinas de la fórmula en la que R1 significa alquilo, en caso dado substituido, alquenilo, en caso dado substituido, alquinilo, en caso dado substituido, cicloalquilo en caso dado substituido, cicloalquenilo, en caso dado substituido o significa heterociclilo en caso dado substituido, R2 significa hidrógeno, halógeno, alquilo, en caso dado substituido o cicloalquilo, en caso dado substituido, R3 significa heterociclilo, en caso dado substituido, G significa oxigeno o SOn, donde n significa 0, 1 o 2, y X significa halógeno, ciano, alquilo, en caso dado substituido, alcoxi, en caso dado substituido, alquiltio, en caso dado substituido, alquilsulfinilo, en caso dado substituido o alquilsulfonilo, en caso dado substituido.2.- Triazolopirimidinas de la fórmula (I), según la reivindicación 1, en las que R1 significa alquilo con 1 hasta 6 átomos de carbono, que puede estar substituido de una a cinco veces, de forma igual o de formas diferentes, por halógeno, por ciano, por alcoxi con 1 hasta 4 átomos de carbono, y/o por cicloalquilo con 3 hasta 6 átomos de carbono, o R1 significa alquenilo con 2 hasta 6 átomos de carbono, que puede estar substituido de una hasta tres veces, de forma igual o de formas diferentes, por halógeno, por ciano, por hidroxi, por alcoxi con 1 hasta 4 átomos de carbono y/o por cicloalquilo con 3 hasta 6 átomos de carbono, o R1 significa alquinilo con 3 hasta 6 átomos de carbono, que puede estar substituido de una hasta tres veces, de forma igual o de formas diferentes, por halógeno, por ciano, por alcoxi con 1 hasta 4 átomos de carbono y/o por cicloalquilo con 3 hasta 6 átomos de carbono, oR1 significa cicloalquilo con 3 hasta 6 átomos de carbono, que puede estar substituido desde una hasta tres veces, de forma igual o de formas diferentes, por halógeno y/o por alquilo con 1 hasta 4 átomos de carbono, o ...

122. 发明专利

CA2590220A1 2-ALKYL-CYCLOALK(EN)YL-CARBOXAMIDES 未知
公开(公告)号：CA2590220A1
公开(公告)日：2006-06-15
申请号：CA2590220
申请日：2005-12-08
申请人： BAYER CROPSCIENCE AG
发明人： ELBE HANS-LUDWIG , SEITZ THOMAS , GREUL JOERG NICO , WACHENDORFF-NEUMANN ULRIKE , DAHMEN PETER , GAYER HERBERT , KUCK KARL-HEINZ , DUNKEL RALF , HARTMANN BENOIT
IPC分类号： C07D277/56 , A01N43/28 , C07C233/00 , C07D207/34 , C07D213/82 , C07D231/14 , C07D241/24 , C07D307/24 , C07D327/06 , C07D333/38 , C07F7/08
摘要： 2-Alkyl-cycloalk(en)yl-carboxamide compounds (I) are new. 2-Alkyl-cycloalk(en)yl-carboxamide compounds (I) of formula (A-CO-N(R 1>)-L-CH 2(R 2>)-(CH 2) s-X) are new. X : -CR 3>R 4>R 5> or -SiR 49>R 50>R 51>; s : 1-2; R 1>H, 1-8C alkyl, 1-6C alkylsulfinyl, 1-6C alkylsulfonyl, 1-4C alkoxy-1-4C-alkyl, 3-8C cycloalkyl, 1-6C haloalkyl, 1-4C haloalkylthio, 1-4C haloalkylsulfinyl, 1-4C haloalkylsulfonyl, halo-1-4C-alkoxy-1-4C-alkyl, 3-8C halocycloalkyl (with 1-9 of F, Cl and/or Br), formyl, formyl-1-3C-alkyl, (1-3C-alkyl)carbonyl-1-3C-alkyl, (1-3C-alkoxy)carbonyl-1-3C-alkyl, halo-(1-3C-alkyl)carbonyl-1-3C-alkyl, halo-(1-3C-alkoxy)carbonyl-1-3C-alkyl (with 1-13 of F, Cl and/or Br), (1-8C-alkyl)carbonyl, (1-8C-alkoxy)carbonyl, (1-4C-alkoxy-1-4C-alkyl)carbonyl, (3-8C-cycloalkyl)carbonyl, (1-6C-haloalkyl)carbonyl, (1-6C-haloalkoxy)carbonyl, (halo-1-4C-alkoxy-1-4C-alkyl)carbonyl, (3-8C-halocycloalkyl)carbonyl (with 1-9 of F, Cl and/or Br), -C(=O)C(=O)R 6>, -CONR 7>R 8> or -CH 2NR 9>R 10>; L : L 1> or L 2>; L 1>3-7C cycloalkyl-1,2-ene (3-7C-cycloalkyl-1,2-diyl) (optionally substituted by 1-4 of F, Cl, 1-4C alkyl or 1-4C haloalkyl); L 2>cyclohexenylene (cyclohexendiyl) (optionally substituted by 1-4 of F, Cl, 1-4C alkyl or 1-4C haloalkyl); R 2>H, halo, 1-4C alkyl or 1-4C haloalkyl with 1-9 of F, Cl and/or Br; either R 3>halo, 1-8C alkyl or 1-6C haloalkyl with 1-13 of F, Cl and/or Br; and R 4>halo, 1-8C alkyl or 1-6C haloalkyl with 1-13 of F, Cl and/or Br; or CR 3>R 4>3-6 membered, optionally unsaturated, carbocyclic or heterocyclic ring (optionally substituted with halo, 1-4C alkyl, 1-4C alkoxy, 1-4C haloalkyl or 1-4C haloalkoxy); R 5>H, halo, 1-8C alkyl or 1-6C haloalkyl with 1-13 of F, Cl and/or Br; R 49>, R 50>H, 1-8C alkyl, 1-8C alkoxy, 1-4C alkoxy-1-4C-alkyl, 1-4C alkylthio-1-4C-alkyl or 1-6C haloalkyl; R 51>phenyl, phenylalkyl (both optionally substituted), H, 1-8C alkyl, 1-8C alkoxy, 1-4C alkoxy-1-4C-alkyl, 1-4C-alkylthio-1-4C-alkyl, 2-8C alkenyl, 2-8C-alkynyl, 1-6C haloalkyl, 2-6C haloalkenyl, 2-6C haloalkynyl or 3-6C cycloalkyl; R 6>H, 1-8C alkyl, 1-8C alkoxy, 1-4C alkoxy-1-4C-alkyl, 3-8C cycloalkyl, 1-6C haloalkyl, 1-6C haloalkoxy, halo-1-4C-alkoxy-1-4C-alkyl or 3-8C-halocycloalkyl with 1-9 of F, Cl and/or Br; either R 7>, R 8>H, 1-8C alkyl, 1-4C alkoxy-1-4C-alkyl, 3-8C cycloalkyl, 1-8C haloalkyl, halo-1-4C-alkoxy-1-4C-alkyl or 3-8C-halocycloalkyl with 1-9 of F, Cl and/or Br; or NR 7>R 8>5-8 membered saturated heterocycle (optionally containing 1-2 further non-adjacent heteroatoms of O, S or NR 11>) optionally substituted with one or more halo or 1-4C alkyl; either R 9>, R 10>H, 1-8C alkyl, 3-8C cycloalkyl, 1-8C haloalkyl or 3-8C-halocycloalkyl with 1-9 of F, Cl and/or Br; or NR 9>R 10>5-8 membered saturated heterocycle (optionally containing 1-2 further non-adjacent heteroatoms of O, S or NR 11>), optionally substituted with halo or 1-4C alkyl; R 11>H or 1-6C alkyl; A : 19 (hetero)cyclic groups e.g. phenyl compound of formula (1), pyridine compound of formula (2) and thio compound of formula (3); R 21>H, halo, OH, CN, 1-6C alkyl; or 1-4C haloalkyl, 1-4C haloalkoxy or 1-4C haloalkylthio, each with 1-5 halo atoms; R 22>H, halo, OH, CN, 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio; or 1-4C haloalkyl, 1-4C haloalkylthio or 1-4C haloalkoxy, each with 1-5 halo atoms; R 23>H, halo, OH, CN, 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio; or 1-4C haloalkyl, 1-4C haloalkoxy, each with1-5 halo atoms, 1-4C-alkylsulfinyl or 1-4C alkylsulfonyl; and R 26>1-4C alkyl or 1-4C haloalkyl with 1-5 halo atoms. Independent claims are also included for: (1) the preparation of (I); (2) agents for combating undesired microorganisms, comprising at least (I) with diluting agent and/or surface active agents; and (3) methods for combating undesired microorganisms, comprising applying (I) with diluting agent and/or surface active agents on the microorganisms and/or its habitat. [Image] ACTIVITY : Antibacterial; Antifungal. MECHANISM OF ACTION : None given.

123. 发明专利

ECSP056201A TRIAZOLOPIRIMIDINAS 未知
公开(公告)号：ECSP056201A
公开(公告)日：2006-04-19
申请号：ECSP056201
申请日：2005-12-02
申请人： BAYER CROPSCIENCE AG
发明人： ELBE HANS LUDWIG , GREUL JOERG NICO , WACHENDORFF-NEUMANN ULRIKE , DAHMEN PETER , KUCK KART-HEINZ , GEBAUER OLAF , HEINEMANN ULRICH , GAYER HERBERT , HERRMANN STEFAN , KRUEGER BERND-WIELAND , HILLEBRAND STEFAN , EBBERT RONALD
IPC分类号： A01N43/90 , C07D213/55 , C07D213/61 , C07D487/04
摘要： Nuevas triazolopirimidinas de la fórmula (I) (I)en la queR1, R2, R3 y X tienen los significados indicados en la descripción, un procedimiento para la obtención de estos productos y su empleo para la lucha contra los microorganismos indeseados. Nuevos productos intermedios (II), (IV), (V-a), (V-b) (II) (IV). (V-a) (V-b)así como procedimientos para la obtención de estos productos.

124. 发明专利

CA2578007A1 BIPHENYL-THIAZOLO-CARBOXAMIDES 未知
公开(公告)号：CA2578007A1
公开(公告)日：2006-03-09
申请号：CA2578007
申请日：2005-08-13
申请人： BAYER CROPSCIENCE AG
发明人： DAHMEN PETER , WACHENDORFF-NEUMANN ULRIKE , SEITZ THOMAS , KUCK KARL-HEINZ , GREUL JOERG NICO , DUNKEL RALF , ELBE HANS-LUDWIG , GAYER HERBERT , HARTMANN BENOIT
IPC分类号： C07D277/56 , A01N43/78
摘要： Novel biphenyl thiazole carboxamides of Formula (I) where R1, R2, R3, R4, R5 and n have the meanings specified in the description, several methods for the manufacture of these substances and their use for combating undesired microorganisms, as well as novel intermediate products and their manufacture.

125. 发明专利

DE102004041530A1 未知
公开(公告)号：DE102004041530A1
公开(公告)日：2006-03-02
申请号：DE102004041530
申请日：2004-08-27
申请人： BAYER CROPSCIENCE AG
发明人： DUNKEL RALF , ELBE HANS-LUDWIG , GREUL JOERG NICO , HARTMANN BENOIT , GAYER HERBERT , SEITZ THOMAS , WACHENDORFF-NEUMANN ULRIKE , DAHMEN PETER , KUCK KARL-HEINZ
IPC分类号： A01N43/78 , C07D277/56 , C07F5/02
摘要： Novel biphenyl thiazole carboxamides of Formula (I) where R1, R2, R3, R4, R5 and n have the meanings specified in the description, several methods for the manufacture of these substances and their use for combating undesired microorganisms, as well as novel intermediate products and their manufacture.

126. 发明专利

ES2238853T3 COMBINACIONES DE PRODUCTOS ACTIVOS FUNGICIDAS. 未知
公开(公告)号：ES2238853T3
公开(公告)日：2005-09-01
申请号：ES99953975
申请日：1999-11-08
申请人： BAYER CROPSCIENCE AG
发明人： MAULER-MACHNIK ASTRID , WACHENDORFF-NEUMANN ULRIKE , GAYER HERBERT
IPC分类号： A01N43/54
摘要： Combinación de productos activos que contiene un compuesto de la fórmula (I), en la que R1 significa hidrógeno, metilo, etilo, metoxi, cloro, bromo, flúor o ciano y El compuesto 1) 1) Spiroxam in en una proporción de mezcla entre un compuesto de la fórmula (I) y el compuesto 1) desde 20:1 hasta 1:50 partes en peso.

127. 发明专利

PL372462A1 TRIAZOLOPYRIMIDINES USED AS FUNGICIDES 未知
公开(公告)号：PL372462A1
公开(公告)日：2005-07-25
申请号：PL37246203
申请日：2003-03-10
申请人： BAYER CROPSCIENCE AG
发明人： BOIE CHRISTIANE , DUNKEL RALF , ELBE HANS-LUDWIG , GAYER HERBERT , GEBAUER OLAF , KRUEGER BERND-WIELAND , HEINEMANN ULRICH , VOERSTE ARND , GUTH OLIVER , EBBERT RONALD , WACHENDORFF-NEUMANN ULRIKE , MAULER-MACHNIK ASTRID
IPC分类号： A01N25/30 , A01N43/90 , C07D249/10 , C07D249/14 , C07D487/04 , A01N43/00
摘要： Novel triazolopyrimidines of the formula in which R 1 represents amino, represents in each case optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkyloxy, alkylamino, dialkylamino, alkenylamino, alkynylamino, cycloalkylamino, N-cycloalkyl-N-alkylamino, alkylideneamino or heterocyclyl, and R 2 represents hydrogen or represents in each case optionally substituted alkyl, alkenyl, alkynyl or cycloalkyl, or R 1 and R 2 together with the nitrogen atom to which they are attached form an optionally substituted heterocyclic ring, R 3 represents aryl which is optionally mono- to tetrasubstituted, R 4 represents halogen, cyano or represents in each case optionally substituted alkoxy or dialkylamino and X represents halogen, a process for preparing these novel substances and their use for controlling unwanted microorganisms. Novel intermediates of the formulae and processes for their preparation.

128. 发明专利

DE10357570A1 New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood 未知
公开(公告)号：DE10357570A1
公开(公告)日：2005-07-07
申请号：DE10357570
申请日：2003-12-10
申请人： BAYER CROPSCIENCE AG
发明人： GEBAUER OLAF , HEINEMANN ULRICH , HERRMANN STEFAN , GUTH OLIVER , ELBE HANS-LUDWIG , GAYER HERBERT , GREUL JOERG NICO , HILLEBRAND STEFAN , EBBERT RONALD , WACHENDORFF-NEUMANN ULRIKE , DAHMEN PETER , KUCK KARL-HEINZ
IPC分类号： A01N43/90 , C07D213/55 , C07D213/61 , C07D487/04
摘要： 3-Substituted 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives (I) are new. Pyrazolo-pyrimidines of formula (I) and their salts are new. [Image] R 1>alkyl, alkenyl, alkynyl, cycloalkyl or heterocyclyl (all optionally substituted); R 2>H or alkyl; or NR 1>R 2>optionally substituted heterocycle; R 3>optionally substituted heterocyclyl; R 4>H or alkyl; Hal : halogen; and X : halo, CN, NO 2, alkyl, optionally substituted alkenyl, optionally substituted alkynyl, hydroxyalkyl, alkylcarbonyl, alkoxyalkyl, haloalkyl, cycloalkyl, CHO, CSNH 2, alkoxycarbonyl, hydroxyiminoalkyl, alkoxyiminoalkyl, alkylthio, alkylsulfinyl, alkylsulfonyl or alkylaminocarbonyl. Independent claims are included for: (a) A method of preparation of (I); (b) Interconversion of (I); (c) New pyrazolo-pyrimidine derivative intermediates of formulae (II) and (X); (d) New pyridyl- or pyrimidinyl-malonate ester derivative intermediates of formulae (XII-a) and (XII-b); and (e) A method of preparation of (II), (X), (XII-a) and (XII-b). [Image] X 1>halo, CN, NO 2, alkyl, haloalkyl, cycloalkyl, CHO, CSNH 2, alkoxycarbonyl, alkylcarbonyl, alkylthio, alkylsulfinyl, alkylsulfonyl or alkylaminocarbonyl; Y 1>halo; R : halo, CN, NO 2, alkyl, haloalkyl, cycloalkyl, CSNH 2, alkoxycarbonyl, alkylthio, alkylsulfinyl, alkylsulfonyl or alkylaminocarbonyl; R 1> 2>1-4C alkyl; R 1> 3>, R 1> 4>halo or haloalkyl; and R 15>, R 1> 6>H, F, CL, Br, Me, Et or OMe. ACTIVITY : Fungicide; antibacterial; algicide; cytostatic; herbicide; plant growth regulator. In tests against Venturia inaequalis in apple tree seedlings, 3-cyano-5-chloro-6-(3-trifluoromethyl-pyridin-2-yl)-pyrazolo-(1,5-a)-pyrimidin-7-yl-N-((1S)-2,2,2-trifluoro-1-methylethyl)-amine (Ia) at an application rate of 100 g/ha gave more than 90% prevention of infection. MECHANISM OF ACTION : None given.

129. 发明专利

DE10357566A1 未知
公开(公告)号：DE10357566A1
公开(公告)日：2005-07-07
申请号：DE10357566
申请日：2003-12-10
申请人： BAYER CROPSCIENCE AG
发明人： GEBAUER OLAF , HEINEMANN ULRICH , HERRMANN STEFAN , GAYER HERBERT , HILLEBRAND STEFAN , ELBE HANS-LUDWIG , EBBERT RONALD , WACHENDORFF-NEUMANN ULRIKE , DAHMEN PETER , KUCK KARL-HEINZ
IPC分类号： A01N43/90 , C07D487/04
摘要： This invention relates to novel pyrazolopyrimidines of the formula in which R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 and R 8 are as defined in the disclosure, to a plurality of processes for preparing these compounds and to their use for controlling unwanted microorganisms.

130. 发明专利

CA2548516A1 PYRAZOLOPYRIMIDINES 未知
公开(公告)号：CA2548516A1
公开(公告)日：2005-06-23
申请号：CA2548516
申请日：2004-12-08
申请人： BAYER CROPSCIENCE AG
发明人： ELBE HANS-LUDWIG , EBBERT RONALD , DAHMEN PETER , GAYER HERBERT , HILLEBRAND STEFAN , GEBAUER OLAF , KUCK KARL-HEINZ , WACHENDORFF-NEUMANN ULRIKE , HEINEMANN ULRICH , HERRMANN STEFAN
IPC分类号： C07D487/04 , A01N43/90 , C07D231/00 , C07D239/00
摘要： Novel pyrazolopyrimidines of formula (I), wherein R1, R2, R3, R4, R5 and R6 have meanings given in the description. Several methods for producing said products and for the use thereof against undesirable microorganisms are also disclosed.

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