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111. 发明授权

US08188295B2 Method for producing difluoromethyl-substituted pyrazole compounds 有权
标题翻译：二氟甲基取代的吡唑化合物的制备方法
公开(公告)号：US08188295B2
公开(公告)日：2012-05-29
申请号：US12664448
申请日：2008-06-13
申请人： Markus Nett , Thomas Grote , Jan Klaas Lohmann , Jochen Dietz , Sebastian Peer Smidt , Michael Rack , Thomas Zierke
发明人： Markus Nett , Thomas Grote , Jan Klaas Lohmann , Jochen Dietz , Sebastian Peer Smidt , Michael Rack , Thomas Zierke
IPC分类号： C07D231/14 , C07C229/06
CPC分类号： C07D231/12 , C07D231/14
摘要： The present invention relates to a process for preparing 3-difluoromethyl-Substituted pyrazole compounds of the formula (I) in which R1 is H, halogen, nitro, C1-C8-alkyl, C1-C8-haloalkyl, C3-C8-cycloalkyl, phenyl, naphthyl, hetaryl, cyano, —C(═O)—OR1a, —C(═O)—NR1bR1c, —C(═O)—SR1d or —C(═S)—SR1e; R2 is H, C1-C4-alkyl, benzyl or phenyl; R3 is H, halogen, C1-C8-alkoxy, C1-C8-haloalkoxy, C3-C8-cycloalkoxy, C2-C8-alkenyloxy, C1-C8-alkylthio, C1-C8-haloalkylthio, C3-C8-cyclo-alkylthio or C2-C8-alkenylthio; compounds of the formula (II.a) or (II.b), in which R1 and R3 each have one of the definitions given above; R4 is halogen, —OR4a, —SR4a, —O—SO2—R4a or an —NR4bR4c group; R5 and R6 are each C1-C8-alkyl, C1-C8-haloalkyl, C3-C8-cycloalkyl, benzyl or phenyl, or, together with the nitrogen atom to which they are bonded, are a 3- to 8-membered heterocycle; Lewis acid adducts of compounds of the formula (II.b); the use of compounds of the formula (II.a) or (II.b) and of the Lewis acid adducts for preparing compounds of the formula (I) or (VI); and to a process for converting such compounds to the corresponding 3-difluoro-pyrazol-4-ylcarboxylic acids.
摘要翻译：本发明涉及一种制备式（I）的3-二氟甲基取代的吡唑化合物的方法，其中R 1是H，卤素，硝基，C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，苯基，萘基，杂芳基，氰基，-C（= O）-OR1a，-C（= O）-NR1bR1c，-C（= O）-SR1d或-C（= S）-SR1e; R2是H，C1-C4-烷基，苄基或苯基; R 3是H，卤素，C 1 -C 8 - 烷氧基，C 1 -C 8 - 卤代烷氧基，C 3 -C 8 - 环烷氧基，C 2 -C 8 - 烯氧基，C 1 -C 8 - 烷硫基，C 1 -C 8 - 卤代烷硫基，C 3 -C 8环 - C 2 -C 8 - 烯硫基; 式（II.a）或（II.b）化合物，其中R 1和R 3各自具有上述定义之一; R4是卤素，-OR4a，-SR4a，-O-SO2-R4a或-NR4bR4c基团; R 5和R 6各自为C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，苄基或苯基，或与它们所键合的氮原子一起为3-至8-元杂环; 式（II.b）化合物的路易斯酸加合物; 使用式（II.a）或（II.b）化合物和路易斯酸加成物制备式（I）或（VI）化合物的方法; 以及将这些化合物转化为相应的3-二氟 - 吡唑-4-基羧酸的方法。

112. 发明授权

US07994340B2 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi, and compositions comprising them 失效
标题翻译：唑基甲基环氧乙烷，它们用于控制植物病原真菌的用途，以及包含它们的组合物
公开(公告)号：US07994340B2
公开(公告)日：2011-08-09
申请号：US12519973
申请日：2007-12-04
申请人： Jens Renner , Thomas Grote , Bernd Müller , Jan Klaas Lohmann , Sarah Ulmschneider , Alice Glättli , Jochen Dietz
发明人： Jens Renner , Thomas Grote , Bernd Müller , Jan Klaas Lohmann , Sarah Ulmschneider , Alice Glättli , Jochen Dietz
IPC分类号： A01N43/64 , C07D249/08
CPC分类号： C07D405/06 , A01N43/653
摘要： The present invention relates to azolylmethyloxiranes of the general formula (I) in which A stands for phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, with the proviso that A does not stand for 2-methylphenyl, and also their plant-compatible acid addition salts or metal salts, and also to the use of the compounds of the formula I for controlling phytopathogenic fungi, and to compositions comprising them.
摘要翻译：本发明涉及通式（I）的唑基甲基环氧乙烷，其中A代表任选被一至三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4 - 烷氧基， C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，条件是A不代表2-甲基苯基，并且还涉及用于控制植物病原真菌的式I化合物以及包含它们的组合物的用途。

113. 发明申请

US20110172098A1 Imidazole and Triazole Compounds, Their Use and Agents Containing the Same 审中-公开
公开(公告)号：US20110172098A1
公开(公告)日：2011-07-14
申请号：US13119969
申请日：2009-09-09
申请人： Jochen Dietz , Thomas Grote , Bernd Müller , Jan Klaas Lohmann , Jens Renner , Sarah Ulmschneider , Alice Glättli , Marianna Vrettou , Wassillos Grammenos
发明人： Jochen Dietz , Thomas Grote , Bernd Müller , Jan Klaas Lohmann , Jens Renner , Sarah Ulmschneider , Alice Glättli , Marianna Vrettou , Wassillos Grammenos
IPC分类号： A01N25/26 , C07D249/08 , A01N43/707 , A01P13/00 , A01P3/00 , A01P7/04
CPC分类号： C07D249/08 , C07D233/60
摘要： The present invention relates to compounds of the formula I in which the variables have the meanings defined in the claims and in the description.

114. 发明申请

US20090305887A1 Azolylmethyloxiranes, Their Use for Controlling Phytopathogenic Fungi and Compositions Comprising Them 审中-公开
标题翻译：唑基甲基环氧乙烷，它们用于控制植物病原真菌和组合物的用途
公开(公告)号：US20090305887A1
公开(公告)日：2009-12-10
申请号：US12306027
申请日：2007-06-20
申请人： Jochen Dietz , Thomas Grote , Bernd Müller , Jan Klaas Lohmann , Jens Renner , Sarah Ulmschneider , Alice Glättli
发明人： Jochen Dietz , Thomas Grote , Bernd Müller , Jan Klaas Lohmann , Jens Renner , Sarah Ulmschneider , Alice Glättli
IPC分类号： A01N25/34 , C07D249/08 , A01N43/653 , A01P3/00
CPC分类号： C07D405/06
摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A is phenyl which is substituted by an F and another substituent selected from the group consisting of Cl, C1-C4-alkyl, C1-C4-haloalkyl and C1-C4-alkoxy, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl or is phenyl which is substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, with the proviso that B is not o-methylphenyl if A is 2-chloro-4-fluorophenyl, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.
摘要翻译：本发明涉及通式I的唑基甲基环氧烷，其中A是被F取代的苯基，另一个选自Cl，C 1 -C 4 - 烷基，C 1 -C 4卤代烷基和C 1 -C 4 - 烷氧基的取代基 B是未取代的吡啶基，噻吩基，噻唑基，恶唑基或呋喃基，或被一至三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，条件是如果A是2-氯-4-氟苯基，则B不是邻甲基苯基，涉及与植物相容的酸加成盐或其金属盐，用于控制植物病原真菌的式I化合物和包含这些化合物的组合物。

115. 发明申请

US20090036305A1 PYRAZOLECARBOXAMIDES 失效
标题翻译：吡咯烷氧基胺
公开(公告)号：US20090036305A1
公开(公告)日：2009-02-05
申请号：US11919588
申请日：2006-05-10
申请人： Markus Gewehr , Jochen Dietz , Thomas Grote , Wassilios Gremmenos , Udo Hunger , Bernd Muller , Frank Schieweck , Anja Schwogler , Jan Klaas Lohmann , Joachim Rheinheimer , Jens Renner , Peter Schafer
发明人： Markus Gewehr , Jochen Dietz , Thomas Grote , Wassilios Gremmenos , Udo Hunger , Bernd Muller , Frank Schieweck , Anja Schwogler , Jan Klaas Lohmann , Joachim Rheinheimer , Jens Renner , Peter Schafer
IPC分类号： A01N43/56 , C07D231/14 , A01P3/00
CPC分类号： A01N43/56 , C07D231/14
摘要： The present invention relates to pyrazolecarboxamides of the formula I in which the variables are as defined below: X is trifluoromethyl; R1 is F, Cl, Br, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen, halogen or C1-C4-alkyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C2-C4-alkynyl or C3-C6-cycloalkyl; W is O or S; with the proviso that, if R3 is hydrogen and W is oxygen, a) R1 and R2 are not simultaneously methyl and F, respectively; b) R1 and R2 are not simultaneously trifluoromethyl and hydrogen or fluorine, respectively. to processes for preparing these compounds, to seeds and compositions comprising them and to methods for controlling harmful fungi.
摘要翻译：本发明涉及式I的吡唑酰胺，其中变量如下所定义：X是三氟甲基; R1是F，Cl，Br，C1-C4-烷基或C1-C4卤代烷基; R2是氢，卤素或C1-C4-烷基; R 3是氢，C 1 -C 4 - 烷基，C 1 -C 4卤代烷基，C 2 -C 4 - 烯基，C 2 -C 4 - 炔基或C 3 -C 6 - 环烷基; W为O或S; 条件是，如果R3是氢并且W是氧，则a）R1和R2分别不同时为甲基和F; b）R1和R2分别不同时为三氟甲基和氢或氟。制备这些化合物的方法，包括它们的种子和组合物以及用于控制有害真菌的方法。

116. 发明申请

US20110319665A1 Process for Preparing Substituted 2-Nitrobiphenyls 有权
标题翻译：制备取代的2-硝基联苯的方法
公开(公告)号：US20110319665A1
公开(公告)日：2011-12-29
申请号：US13254946
申请日：2010-03-08
申请人： Alexander Korte , Jan Klaas Lohmann , Thomas Grote , Klaus Ebel , Thomas Zierke , Horst Mayer , Ralf Wazulek
发明人： Alexander Korte , Jan Klaas Lohmann , Thomas Grote , Klaus Ebel , Thomas Zierke , Horst Mayer , Ralf Wazulek
IPC分类号： C07C205/06 , C07C211/52
CPC分类号： C07C205/11 , C07C205/09 , C07C205/10 , C07C2601/16
摘要： The present invention relates to a process for preparing substituted 2-nitrobiphenyls and to specific 2-nitrobiphenyls. The invention further relates to a process for preparing 2-aminobiphenyls from such 2-nitrobiphenyls and to a process for preparing (het)arylamides of such 2-aminobiphenyls.
摘要翻译：本发明涉及制备取代的2-硝基联苯和特定2-硝基联苯的方法。本发明还涉及从这种2-硝基联苯制备2-氨基联苯的方法和制备这种2-氨基联苯的（het）芳基酰胺的方法。

117. 发明授权

US08853455B2 Process for preparing substituted 2-nitrobiphenyls 有权
标题翻译：制备取代的2-硝基联苯的方法
公开(公告)号：US08853455B2
公开(公告)日：2014-10-07
申请号：US13254946
申请日：2010-03-08
申请人： Alexander Korte , Jan Klaas Lohmann , Thomas Grote , Klaus Ebel , Thomas Zierke , Horst Mayer , Ralf Wazulek
发明人： Alexander Korte , Jan Klaas Lohmann , Thomas Grote , Klaus Ebel , Thomas Zierke , Horst Mayer , Ralf Wazulek
IPC分类号： C07C211/00 , C07C209/00 , C07C205/11 , C07C205/10 , C07C205/09
CPC分类号： C07C205/11 , C07C205/09 , C07C205/10 , C07C2601/16
摘要： The present invention relates to a process for preparing substituted 2-nitrobiphenyls and to specific 2-nitrobiphenyls. The invention further relates to a process for preparing 2-aminobiphenyls from such 2-nitrobiphenyls and to a process for preparing (het)arylamides of such 2-aminobiphenyls.
摘要翻译：本发明涉及制备取代的2-硝基联苯和特定2-硝基联苯的方法。本发明还涉及从这种2-硝基联苯制备2-氨基联苯的方法和制备这种2-氨基联苯的（het）芳基酰胺的方法。

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