发明申请
WO2022199661A1 PHENYL- [1, 3] DIOXOLO [4, 5-C] PYRIDINYL-PHENYL-, PHENYL- [1, 3] DIOXOLO [4, 5-C] PYRIDINYL-HETEROARYL-, OR PHENYL- [1, 3] DIOXOLO [4, 5-C] PYRIDINYL-PIPERIDINYL-METHYL-OXETANYLMETHYL-1H-BENZO [D] IMIDAZOLE-CARBOXYLIC ACID DERIVATIVES AND METHODS OF USING SAME
审中-公开
基本信息:
- 专利标题: PHENYL- [1, 3] DIOXOLO [4, 5-C] PYRIDINYL-PHENYL-, PHENYL- [1, 3] DIOXOLO [4, 5-C] PYRIDINYL-HETEROARYL-, OR PHENYL- [1, 3] DIOXOLO [4, 5-C] PYRIDINYL-PIPERIDINYL-METHYL-OXETANYLMETHYL-1H-BENZO [D] IMIDAZOLE-CARBOXYLIC ACID DERIVATIVES AND METHODS OF USING SAME
- 申请号:PCT/CN2022/082788 申请日:2022-03-24
- 公开(公告)号:WO2022199661A1 公开(公告)日:2022-09-29
- 发明人: REN, Zaifang , SUN, Xuefeng , ZHOU, Jingye
- 申请人: ECCOGENE (SHANGHAI) CO., LTD.
- 申请人地址: Room 402A, Aidisheng Road 326, Pudong
- 专利权人: ECCOGENE (SHANGHAI) CO., LTD.
- 当前专利权人: ECCOGENE (SHANGHAI) CO., LTD.
- 当前专利权人地址: Room 402A, Aidisheng Road 326, Pudong
- 代理机构: AFD CHINA INTELLECTUAL PROPERTY LAW OFFICE
- 优先权: CNPCT/CN2021/082781 2021-03-24
- 主分类号: C07D401/04
- IPC分类号: C07D401/04 ; C07D405/04 ; C07D417/14 ; C07D487/04 ; A61K31/497 ; A61P3/10
摘要:
Provided is compound of Formula (Y) or Formula (A) or pharmaceutically acceptable salt, hydrate, solvate, prodrug, stereoisomer, or tautomer thereof, which modulates the activity of GLP-1 receptor, a pharmaceutical composition comprising a compound of Formula (I), and a method of treating or preventing a disease in which GLP-1 receptor plays a role.
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D401/00 | 杂环化合物,含有两个或更多个杂环,以氮原子作为仅有的杂环原子,至少有1个环是仅含有1个氮原子的六元环 |
--------C07D401/02 | .含有两个杂环 |
----------C07D401/04 | ..被环原子—环原子的键直接连接的 |