基本信息:
- 专利标题: INSULIN RECEPTOR PARTIAL AGONISTS
- 申请号:PCT/US2021/047304 申请日:2021-08-24
- 公开(公告)号:WO2022046739A1 公开(公告)日:2022-03-03
- 发明人: MADSEN-DUGGAN, Christina, B. , FENG, Danqing , HUO, Pei , KEKEC, Ahmet , LIN, Songnian , NARGUND, Ravi , MOYES, Christopher, R. , PISSARNITSKI, Dmitri, A. , SHI, Zhicai , WU, Zhicai , YAN, Lin , ZHU, Yuping
- 申请人: MERCK SHARP & DOHME CORP. , MADSEN-DUGGAN, Christina, B. , FENG, Danqing , HUO, Pei , KEKEC, Ahmet , LIN, Songnian , NARGUND, Ravi , MOYES, Christopher, R. , PISSARNITSKI, Dmitri, A. , SHI, Zhicai , WU, Zhicai , YAN, Lin , ZHU, Yuping
- 申请人地址: 126 East Lincoln Avenue; 805 Muir Terrace; 2000 Galloping Hill Road; 2000 Galloping Hill Road; 2000 Galloping Hill Road; 2000 Galloping Hill Road; 12 Coldstream Court; 232 Clifton Street; 2000 Galloping Hill Road; 50 Monica Way; 2000 Galloping Hill Road; 4 Schindler Court; 2000 Galloping Hill Road
- 专利权人: MERCK SHARP & DOHME CORP.,MADSEN-DUGGAN, Christina, B.,FENG, Danqing,HUO, Pei,KEKEC, Ahmet,LIN, Songnian,NARGUND, Ravi,MOYES, Christopher, R.,PISSARNITSKI, Dmitri, A.,SHI, Zhicai,WU, Zhicai,YAN, Lin,ZHU, Yuping
- 当前专利权人: MERCK SHARP & DOHME CORP.,MADSEN-DUGGAN, Christina, B.,FENG, Danqing,HUO, Pei,KEKEC, Ahmet,LIN, Songnian,NARGUND, Ravi,MOYES, Christopher, R.,PISSARNITSKI, Dmitri, A.,SHI, Zhicai,WU, Zhicai,YAN, Lin,ZHU, Yuping
- 当前专利权人地址: 126 East Lincoln Avenue; 805 Muir Terrace; 2000 Galloping Hill Road; 2000 Galloping Hill Road; 2000 Galloping Hill Road; 2000 Galloping Hill Road; 12 Coldstream Court; 232 Clifton Street; 2000 Galloping Hill Road; 50 Monica Way; 2000 Galloping Hill Road; 4 Schindler Court; 2000 Galloping Hill Road
- 代理机构: MERCK SHARP & DOHME CORP.
- 优先权: US63/070,384 2020-08-26
- 主分类号: C07K14/62
- IPC分类号: C07K14/62 ; A61P3/10
摘要:
Insulin dimers and insulin analog dimers that act as partial agonists at the insulin receptor are disclosed.