基本信息:
- 专利标题: COMPOUNDS USEFUL FOR INHIBITING ROR-GAMMA-T
- 申请号:PCT/US2018/019920 申请日:2018-02-27
- 公开(公告)号:WO2018160550A1 公开(公告)日:2018-09-07
- 发明人: CLARKE, Christian Alexander , LUGAR III, Charles Willis , MORPHY, John Richard , RICHARDSON, Timothy Ivo , RUDYK, Helene , SAPMAZ, Selma , STITES, Ryan Edward , VAUGHT, Grant Mathews
- 申请人: ELI LILLY AND COMPANY
- 申请人地址: Lilly Corporate Center Indianapolis, Indiana 46285 US
- 专利权人: ELI LILLY AND COMPANY
- 当前专利权人: ELI LILLY AND COMPANY
- 当前专利权人地址: Lilly Corporate Center Indianapolis, Indiana 46285 US
- 代理机构: DINGESS-HAMMOND, Elizabeth A. et al.
- 优先权: US62/466,117 20170302
- 主分类号: C07D495/20
- IPC分类号: C07D495/20 ; A61P37/02 ; A61P29/00 ; A61K31/438
摘要:
The present invention provides novel ROR gamma-t inhibitors and pharmaceutical compositions thereof, formula (A).
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D495/00 | 杂环化合物,在稠环系中至少有1个杂环具有硫原子作为仅有的杂环原子 |
--------C07D495/02 | .在稠环系中含有两个杂环 |
----------C07D495/20 | ..螺稠合系 |