基本信息:
- 专利标题: BIPARATOPIC BINDING POLYPEPTIDES FOR CXCR2 AND USES THEREOF
- 专利标题(中):用于CXCR2的双相结合聚合物及其用途
- 申请号:PCT/IB2013053711 申请日:2013-05-08
- 公开(公告)号:WO2013168108A3 公开(公告)日:2014-02-13
- 发明人: BROWN ZARIN , BRADLEY MICHELLE , CHARLTON STEVEN JOHN , VAN HEEKE GINO ANSELMUS , CROMIE KAREN , DOMBRECHT BRUNO , STEFFENSEN SOREN , BAUMEISTER JUDITH , BOUCHE MARIE-PAULE , BOUTTON CARLO , BUYSE MARIE-ANGE , SNOECK VEERLE , STAELENS STEPHANIE
- 申请人: NOVARTIS AG , BROWN ZARIN , BRADLEY MICHELLE , CHARLTON STEVEN JOHN , VAN HEEKE GINO ANSELMUS , CROMIE KAREN , DOMBRECHT BRUNO , STEFFENSEN SOREN , BAUMEISTER JUDITH , BOUCHE MARIE-PAULE , BOUTTON CARLO , BUYSE MARIE-ANGE , SNOECK VEERLE , STAELENS STEPHANIE
- 专利权人: NOVARTIS AG,BROWN ZARIN,BRADLEY MICHELLE,CHARLTON STEVEN JOHN,VAN HEEKE GINO ANSELMUS,CROMIE KAREN,DOMBRECHT BRUNO,STEFFENSEN SOREN,BAUMEISTER JUDITH,BOUCHE MARIE-PAULE,BOUTTON CARLO,BUYSE MARIE-ANGE,SNOECK VEERLE,STAELENS STEPHANIE
- 当前专利权人: NOVARTIS AG,BROWN ZARIN,BRADLEY MICHELLE,CHARLTON STEVEN JOHN,VAN HEEKE GINO ANSELMUS,CROMIE KAREN,DOMBRECHT BRUNO,STEFFENSEN SOREN,BAUMEISTER JUDITH,BOUCHE MARIE-PAULE,BOUTTON CARLO,BUYSE MARIE-ANGE,SNOECK VEERLE,STAELENS STEPHANIE
- 优先权: US201261644582 2012-05-09
- 主分类号: C07K16/28
- IPC分类号: C07K16/28
摘要:
The present invention relates to polypeptides directed against or specifically binding to chemokine receptor CXCR2 and in particular to polypeptides capable of modulating signal transduction from CXCR2. The invention also relates to nucleic acids, vectors and host cells capable of expressing the polypeptides of the invention, pharmaceutical compositions comprising the polypeptides and uses of said polypeptides and compositions for treatment of diseases involving aberrant functioning of CXCR2.
摘要(中):
本发明涉及针对或特异性结合趋化因子受体CXCR2的多肽,特别涉及能够调节CXCR2信号转导的多肽。 本发明还涉及能够表达本发明多肽的核酸,载体和宿主细胞,包含多肽的药物组合物以及用于治疗涉及CXCR2异常功能的疾病的所述多肽和组合物的用途。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07K | 肽 |
------C07K16/00 | 免疫球蛋白,例如,单克隆或多克隆抗体 |
--------C07K16/18 | .来自动物或人的抵抗物质 |
----------C07K16/28 | ..抗受体,细胞表面抗原或细胞表面决定因子 |