基本信息:
- 专利标题: BROMODOMAIN INHIBITORS
- 专利标题(中):BROMODOMAIN抑制剂
- 申请号:PCT/CN2012/086357 申请日:2012-12-11
- 公开(公告)号:WO2013097601A1 公开(公告)日:2013-07-04
- 发明人: WANG, Le , PRATT, John K. , MCDANIEL, Keith F. , DAI, Yujia , FIDANZE, Steven D. , HASVOLD, Lisa , HOLMS, James H. , KATI, Warren M. , LIU, Dachun , MANTEI, Robert A. , MCCLELLAN, William J , SHEPPARD, George S. , WADA, Carol K.
- 申请人: ABBVIE INC. , ABBOTT LABORATORIES TRADING (SHANGHAI) COMPANY, LTD.
- 申请人地址: 1 North Waukegan Road North Chicago Illinois 60064 US
- 专利权人: ABBVIE INC.,ABBOTT LABORATORIES TRADING (SHANGHAI) COMPANY, LTD.
- 当前专利权人: ABBVIE INC.,ABBOTT LABORATORIES TRADING (SHANGHAI) COMPANY, LTD.
- 当前专利权人地址: 1 North Waukegan Road North Chicago Illinois 60064 US
- 代理机构: CHINA PATENT AGENT (HK) LTD.
- 优先权: CNPCT/CN2011/002224 20111230
- 主分类号: C07D471/04
- IPC分类号: C07D471/04 ; A61K31/407 ; A61P35/00 ; A61P31/18 ; A61P13/12 ; A61P3/10
摘要:
The present invention provides for compounds of formula (I) wherein A 1 , A 2 , A 3 , A 4 , X 1 , X 2 , Y 1 , L 1 , G 1 , R x , and R y have any of the values defined thereof in the specification, and pharmaceutically acceptable salts thereof, that are useful as agents in the treatment of diseases and conditions, including inflammatory diseases, cancer, and AIDS. Also provided are pharmaceutical compositions comprising one or more compounds of formula (I).
摘要(中):
本发明提供式(I)化合物,其中A1,A2,A3,A4,X1,X2,Y1,L1,G1,Rx和Ry具有说明书中定义的任何值及其药学上可接受的盐 ,其作为治疗疾病和病症(包括炎性疾病,癌症和AIDS)的药剂是有用的。 还提供了包含一种或多种式(I)化合物的药物组合物。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D471/00 | 在稠环系中含有氮原子作为仅有的杂环原子、其中至少1个环是含有1个氮原子的六元环的杂环化合物,C07D451/00至C07D463/00不包括的 |
--------C07D471/02 | .在稠环系中含两个杂环 |
----------C07D471/04 | ..邻位稠环系 |