基本信息:
- 专利标题: BICYCLIC ACETYL-COA CARBOXYLASE INHIBITORS
- 专利标题(中):双酚A乙酰羧化酶抑制剂
- 申请号:PCT/EP2011/062933 申请日:2011-07-27
- 公开(公告)号:WO2012013716A1 公开(公告)日:2012-02-02
- 发明人: BARNES, David, Weninger , BEBERNITZ, Gregory, Raymond , CLAIRMONT, Kevin , COHEN, Scott, Louis , DAMON, Robert, Edson, II. , DAY, Robert, Francis , DODD, Stephanie, Kay , GAUL, Christoph , GULGEZE EFTHYMIOU, Hatice, Belgin , JAIN, Monish , KARKI, Rajeshri Ganesh , KIRMAN, Louise, Clare , LIN, Kai , MAO, Justin Yik Ching , PATEL, Tajesh Jayprakash , RAYMER, Brian, Kenneth , SU, Liansheng
- 申请人: NOVARTIS AG , BARNES, David, Weninger , BEBERNITZ, Gregory, Raymond , CLAIRMONT, Kevin , COHEN, Scott, Louis , DAMON, Robert, Edson, II. , DAY, Robert, Francis , DODD, Stephanie, Kay , GAUL, Christoph , GULGEZE EFTHYMIOU, Hatice, Belgin , JAIN, Monish , KARKI, Rajeshri Ganesh , KIRMAN, Louise, Clare , LIN, Kai , MAO, Justin Yik Ching , PATEL, Tajesh Jayprakash , RAYMER, Brian, Kenneth , SU, Liansheng
- 申请人地址: Lichtstrasse 35 CH-4056 Basel CH
- 专利权人: NOVARTIS AG,BARNES, David, Weninger,BEBERNITZ, Gregory, Raymond,CLAIRMONT, Kevin,COHEN, Scott, Louis,DAMON, Robert, Edson, II.,DAY, Robert, Francis,DODD, Stephanie, Kay,GAUL, Christoph,GULGEZE EFTHYMIOU, Hatice, Belgin,JAIN, Monish,KARKI, Rajeshri Ganesh,KIRMAN, Louise, Clare,LIN, Kai,MAO, Justin Yik Ching,PATEL, Tajesh Jayprakash,RAYMER, Brian, Kenneth,SU, Liansheng
- 当前专利权人: NOVARTIS AG,BARNES, David, Weninger,BEBERNITZ, Gregory, Raymond,CLAIRMONT, Kevin,COHEN, Scott, Louis,DAMON, Robert, Edson, II.,DAY, Robert, Francis,DODD, Stephanie, Kay,GAUL, Christoph,GULGEZE EFTHYMIOU, Hatice, Belgin,JAIN, Monish,KARKI, Rajeshri Ganesh,KIRMAN, Louise, Clare,LIN, Kai,MAO, Justin Yik Ching,PATEL, Tajesh Jayprakash,RAYMER, Brian, Kenneth,SU, Liansheng
- 当前专利权人地址: Lichtstrasse 35 CH-4056 Basel CH
- 代理机构: CAMPBELL, Lachlan
- 优先权: US61/368,820 20100729
- 主分类号: C07D215/36
- IPC分类号: C07D215/36 ; C07D235/18 ; C07D401/04 ; C07D401/12 ; C07D403/04 ; C07D405/04 ; C07D413/12 ; C07D471/04 ; C07D513/04 ; C07D263/57 ; A61K31/404 ; A61K31/4184
摘要:
The present invention provides compounds of formula (I); or pharmaceutically acceptable salts thereof, wherein the variables are defined as herein. The present invention provides a method for manufacturing the compounds of formula (I), their therapeutic uses, combinations with other of pharmacologically active agents, and a pharmaceutical compositions.
摘要(中):
本发明提供式(I)化合物; 或其药学上可接受的盐,其中变量如本文所定义。 本发明提供了制备式(I)化合物,其治疗用途,与其他药理活性剂的组合以及药物组合物的方法。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D215/00 | 杂环化合物,含喹啉或氢化喹啉环系 |
--------C07D215/02 | .环氮原子和非环原子间无键或只有氢原子或碳原子直接连在环氮原子上 |
----------C07D215/04 | ..只有氢原子或仅含氢和碳原子的基直接连在环碳原子上 |
------------C07D215/36 | ...硫原子 |