基本信息:
- 专利标题: CRTH2 MODULATORS
- 专利标题(中):CRTH2调制器
- 申请号:PCT/US2011/041772 申请日:2011-06-24
- 公开(公告)号:WO2012009134A1 公开(公告)日:2012-01-19
- 发明人: BARDEN, Timothy , HUDSON, Colleen , JIA, James , KIM, Charles , GRAUL, Regina , MERMERIAN, Ara , MOORE, Joel , SPROTT, Kevin , CHIEN, Yueh-tyng
- 申请人: IRONWOOD PHARMACEUTICALS, INC. , BARDEN, Timothy , HUDSON, Colleen , JIA, James , KIM, Charles , GRAUL, Regina , MERMERIAN, Ara , MOORE, Joel , SPROTT, Kevin , CHIEN, Yueh-tyng
- 申请人地址: 301 Binney Street, 2nd Floor Cambridge, MA 02142 US
- 专利权人: IRONWOOD PHARMACEUTICALS, INC.,BARDEN, Timothy,HUDSON, Colleen,JIA, James,KIM, Charles,GRAUL, Regina,MERMERIAN, Ara,MOORE, Joel,SPROTT, Kevin,CHIEN, Yueh-tyng
- 当前专利权人: IRONWOOD PHARMACEUTICALS, INC.,BARDEN, Timothy,HUDSON, Colleen,JIA, James,KIM, Charles,GRAUL, Regina,MERMERIAN, Ara,MOORE, Joel,SPROTT, Kevin,CHIEN, Yueh-tyng
- 当前专利权人地址: 301 Binney Street, 2nd Floor Cambridge, MA 02142 US
- 代理机构: WONG, King, L. et al.
- 优先权: US61/363,501 20100712
- 主分类号: C07D209/10
- IPC分类号: C07D209/10 ; C07D401/06 ; C07D403/06 ; C07D409/06 ; C07D471/04 ; C07D493/04 ; A61K31/404 ; A61P31/06 ; A61P17/00
摘要:
Modulators of CRTH2, particularly antagonists of CRTH2, that are useful for treating various disorders, including asthma and respiratory disorders are disclosed. The compounds fall within a genus described by Formula I:
摘要(中):
公开了可用于治疗各种疾病(包括哮喘和呼吸系统疾病)的CRTH2调节剂,特别是CRTH2拮抗剂。 化合物属于由式I描述的属:
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D209/00 | 杂环化合物,含五元环、与其他环稠合、带1个氮原子作为惟一的杂环原子 |
--------C07D209/02 | .与一个碳环稠合 |
----------C07D209/04 | ..吲哚;氢化吲哚 |
------------C07D209/10 | ...有被杂原子取代的烃基,直接连在杂环的碳原子上 |