发明申请
WO2011019538A1 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT
审中-公开
基本信息:
- 专利标题: SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT
- 专利标题(中):取代的环丙基化合物,包含这些化合物的组合物和处理方法
- 申请号:PCT/US2010/044181 申请日:2010-08-03
- 公开(公告)号:WO2011019538A1 公开(公告)日:2011-02-17
- 发明人: WOOD, Harold, B. , ADAMS, Alan, D. , SZEWCZYK, Jason, W. , ZHANG, Yong , YANG, Meng
- 申请人: MERCK SHARP & DOHME CORP. , WOOD, Harold, B. , ADAMS, Alan, D. , SZEWCZYK, Jason, W. , ZHANG, Yong , YANG, Meng
- 申请人地址: 126 East Lincoln Avenue Rahway, New Jersey 07065-0907 US
- 专利权人: MERCK SHARP & DOHME CORP.,WOOD, Harold, B.,ADAMS, Alan, D.,SZEWCZYK, Jason, W.,ZHANG, Yong,YANG, Meng
- 当前专利权人: MERCK SHARP & DOHME CORP.,WOOD, Harold, B.,ADAMS, Alan, D.,SZEWCZYK, Jason, W.,ZHANG, Yong,YANG, Meng
- 当前专利权人地址: 126 East Lincoln Avenue Rahway, New Jersey 07065-0907 US
- 代理机构: MERCK SHARP & DOHME CORP.
- 优先权: US61/233,690 20090813
- 主分类号: A01N43/40
- IPC分类号: A01N43/40 ; A61K31/445
摘要:
Substituted cyclopropyl compounds of the formula I: are disclosed as useful for treating or preventing type 2 diabetes and similar conditions. Pharmaceutically acceptable salts are included as well. The compounds are useful as agonists of the g-protein coupled receptor GPR-119.
摘要(中):
式I的取代的环丙基化合物被公开用于治疗或预防2型糖尿病和类似病症。 也包括药学上可接受的盐。 该化合物可用作g-蛋白偶联受体GPR-119的激动剂。