基本信息:
- 专利标题: POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS
- 专利标题(中):赖氨酸磷酸受体的多环酸拮抗剂
- 申请号:PCT/US2010037316 申请日:2010-06-03
- 公开(公告)号:WO2010141768A3 公开(公告)日:2011-03-31
- 发明人: HUTCHINSON JOHN HOWARD , SEIDERS THOMAS JON , ZHAO LUCY , WANG BOWEI , ARRUDA JEANNIE M , ROPPE JEFFREY ROGER , PARR TIMOTHY , STOCK NICHOLAS SIMON
- 申请人: AMIRA PHARMACEUTICALS INC , HUTCHINSON JOHN HOWARD , SEIDERS THOMAS JON , ZHAO LUCY , WANG BOWEI , ARRUDA JEANNIE M , ROPPE JEFFREY ROGER , PARR TIMOTHY , STOCK NICHOLAS SIMON
- 专利权人: AMIRA PHARMACEUTICALS INC,HUTCHINSON JOHN HOWARD,SEIDERS THOMAS JON,ZHAO LUCY,WANG BOWEI,ARRUDA JEANNIE M,ROPPE JEFFREY ROGER,PARR TIMOTHY,STOCK NICHOLAS SIMON
- 当前专利权人: AMIRA PHARMACEUTICALS INC,HUTCHINSON JOHN HOWARD,SEIDERS THOMAS JON,ZHAO LUCY,WANG BOWEI,ARRUDA JEANNIE M,ROPPE JEFFREY ROGER,PARR TIMOTHY,STOCK NICHOLAS SIMON
- 优先权: US18378509 2009-06-03
- 主分类号: C07D413/04
- IPC分类号: C07D413/04 ; A61K31/42 ; A61P11/00 ; C07D261/14
摘要:
Described herein are compounds that are antagonists of lysophosphatidic receptor(s). Also described are pharmaceutical compositions and medicaments that include the compounds described herein, as well as methods of using such antagonists, alone and in combination with other compounds, for treating LPA-dependent or LPA-mediated conditions or diseases.
摘要(中):
本文描述的是作为溶血磷脂受体拮抗剂的化合物。 还描述了包括本文所述化合物的药物组合物和药物,以及使用这些拮抗剂单独和与其它化合物组合用于治疗LPA依赖性或LPA介导的病症或疾病的方法。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D413/00 | 杂环化合物,含两个或更多个杂环,至少有1个环有氮原子和氧原子作为仅有的杂环原子 |
--------C07D413/02 | .含两个杂环 |
----------C07D413/04 | ..被环原子—环原子的键直接连接的 |