基本信息:
- 专利标题: COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS
- 专利标题(中):用于治疗炎症性疾病的化合物
- 申请号:PCT/US2009057798 申请日:2009-09-22
- 公开(公告)号:WO2010036638A3 公开(公告)日:2010-05-27
- 发明人: SHANKAR BANDARPALLE B , KIM SEONG HEON , YU WENSHENG , TONG LING , WONG MICHAEL K C , LAVEY BRIAN J , KOZLOWSKI JOSEPH A , CHEN LEI , RIZVI RAZIA K , KOSINSKI ANETA MARIA , YANG DE-YI , ZHOU GUOWEI , ROSNER KRISTEN E , FIRE LUKE , RICHARD JUDSON E , LI DANSU
- 申请人: SCHERING CORP , SHANKAR BANDARPALLE B , KIM SEONG HEON , YU WENSHENG , TONG LING , WONG MICHAEL K C , LAVEY BRIAN J , KOZLOWSKI JOSEPH A , CHEN LEI , RIZVI RAZIA K , KOSINSKI ANETA MARIA , YANG DE-YI , ZHOU GUOWEI , ROSNER KRISTEN E , FIRE LUKE , RICHARD JUDSON E , LI DANSU
- 专利权人: SCHERING CORP,SHANKAR BANDARPALLE B,KIM SEONG HEON,YU WENSHENG,TONG LING,WONG MICHAEL K C,LAVEY BRIAN J,KOZLOWSKI JOSEPH A,CHEN LEI,RIZVI RAZIA K,KOSINSKI ANETA MARIA,YANG DE-YI,ZHOU GUOWEI,ROSNER KRISTEN E,FIRE LUKE,RICHARD JUDSON E,LI DANSU
- 当前专利权人: SCHERING CORP,SHANKAR BANDARPALLE B,KIM SEONG HEON,YU WENSHENG,TONG LING,WONG MICHAEL K C,LAVEY BRIAN J,KOZLOWSKI JOSEPH A,CHEN LEI,RIZVI RAZIA K,KOSINSKI ANETA MARIA,YANG DE-YI,ZHOU GUOWEI,ROSNER KRISTEN E,FIRE LUKE,RICHARD JUDSON E,LI DANSU
- 优先权: US9968608 2008-09-24
- 主分类号: C07D403/06
- IPC分类号: C07D403/06 ; A61K31/33 ; A61P19/00 ; C07D403/14 ; C07D405/14 ; C07D491/048
摘要:
This invention relates to compounds of the Formula (I) as described herein, or a pharmaceutically acceptable salt, solvate or ester thereof, which can be useful for the treatment of diseases or conditions mediated by MMPs, ADAMs, TACE, aggrecanase, TNF- or combinations thereof.
摘要(中):
本发明涉及本文所述的式(I)化合物或其药学上可接受的盐,溶剂化物或酯,其可用于治疗由MMP,ADAM,TACE,聚集蛋白聚糖蛋白酶,TNF-或介导的疾病或病症 其组合。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D403/00 | 杂环化合物,含有两个或更多的杂环,以氮原子作为仅有的杂环原子,C07D401/00组不包含的 |
--------C07D403/02 | .含两个杂环 |
----------C07D403/06 | ..被仅含脂族碳原子的碳链连接的 |