发明申请
WO2009151299A3 STYRYLBENZOFURAN DERIVATIVES AS INHIBITORS FOR BETA-AMYLOID FIBRIL FORMATION AND PREPARATION METHOD THEREOF
审中-公开
基本信息:
- 专利标题: STYRYLBENZOFURAN DERIVATIVES AS INHIBITORS FOR BETA-AMYLOID FIBRIL FORMATION AND PREPARATION METHOD THEREOF
- 专利标题(中):作为抗坏血酸纤维素形成的抑制剂的苯乙烯苯并呋喃衍生物及其制备方法
- 申请号:PCT/KR2009003165 申请日:2009-06-12
- 公开(公告)号:WO2009151299A3 公开(公告)日:2010-04-01
- 发明人: KIM DONG JIN , YOO KYUNG HO , BYUN JI HUN , KIM YOUNGSOO , KIM HYE YUN , LEE GWAN SUN , KIM MAENG SUP , AHN YOUNG GIL , LEE JI HOON , LEE MYOUNG-HWAN , HWANG HANA , RYU JIYEON
- 申请人: KOREA INST SCI & TECH , HANMI PHARM IND CO LTD , KIM DONG JIN , YOO KYUNG HO , BYUN JI HUN , KIM YOUNGSOO , KIM HYE YUN , LEE GWAN SUN , KIM MAENG SUP , AHN YOUNG GIL , LEE JI HOON , LEE MYOUNG-HWAN , HWANG HANA , RYU JIYEON
- 专利权人: KOREA INST SCI & TECH,HANMI PHARM IND CO LTD,KIM DONG JIN,YOO KYUNG HO,BYUN JI HUN,KIM YOUNGSOO,KIM HYE YUN,LEE GWAN SUN,KIM MAENG SUP,AHN YOUNG GIL,LEE JI HOON,LEE MYOUNG-HWAN,HWANG HANA,RYU JIYEON
- 当前专利权人: KOREA INST SCI & TECH,HANMI PHARM IND CO LTD,KIM DONG JIN,YOO KYUNG HO,BYUN JI HUN,KIM YOUNGSOO,KIM HYE YUN,LEE GWAN SUN,KIM MAENG SUP,AHN YOUNG GIL,LEE JI HOON,LEE MYOUNG-HWAN,HWANG HANA,RYU JIYEON
- 优先权: KR20080055307 2008-06-12
- 主分类号: C07D307/78
- IPC分类号: C07D307/78 ; A61K31/343
摘要:
The present invention relates to a novel compound which efficiently inhibits the formation of beta-amyloid fibrils in the brain to be useful for preventing or treating a degenerative brain disease, a method for preparing same, and a pharmaceutical composition comprising same as an active ingredient.
摘要(中):
本发明涉及有效抑制脑中β-淀粉样蛋白原纤维形成以用于预防或治疗退行性脑病的新型化合物,其制备方法和含有该组合物作为活性成分的药物组合物。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D307/00 | 杂环化合物,含五元环,含有1个氧原子作为仅有的杂环原子 |
--------C07D307/02 | .不和其他环稠合 |
----------C07D307/78 | ..苯并 |