基本信息:
- 专利标题: COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING DISEASES
- 专利标题(中):化合物,组合物和治疗或预防疾病的方法
- 申请号:PCT/US2008/074444 申请日:2008-08-27
- 公开(公告)号:WO2009105123A1 公开(公告)日:2009-08-27
- 发明人: DANISHEFSKY, Samuel, J. , CHOU, Ting-chao , LEI, Xiaoguang
- 申请人: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK , DANISHEFSKY, Samuel, J. , CHOU, Ting-chao , LEI, Xiaoguang
- 申请人地址: 412 Low Memorial Library 535 West 116th Street New York, NY 10027 US
- 专利权人: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK,DANISHEFSKY, Samuel, J.,CHOU, Ting-chao,LEI, Xiaoguang
- 当前专利权人: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK,DANISHEFSKY, Samuel, J.,CHOU, Ting-chao,LEI, Xiaoguang
- 当前专利权人地址: 412 Low Memorial Library 535 West 116th Street New York, NY 10027 US
- 代理机构: MCMURRY, Scott, A. et al.
- 优先权: USUS08/054737 20080222
- 主分类号: A01N43/26
- IPC分类号: A01N43/26 ; A61K31/335
摘要:
The present invention provides compounds of Formula (I), compositions comprising an effective amount of a Compound of Formula (I), optionally with a tubulin-binding drug, methods of their use for treating or preventing cancer or a neurotrophic disorder, inducing a chemoprotective phase II enzyme, DNA, or protein synthesis, enhancing the immune system, and methods for making Compounds of the invention.
摘要(中):
本发明提供式(I)化合物,包含有效量的式(I)化合物,任选地与微管蛋白结合药物的组合物,其用于治疗或预防癌症或神经营养障碍的方法,诱导化学保护作用 II期酶,DNA或蛋白质合成,增强免疫系统以及制备本发明化合物的方法。