基本信息:
- 专利标题: HETEROARYL-SUBSTITUTED PIPERIDINES
- 专利标题(中):杂芳基取代的哌啶
- 申请号:PCT/EP2008009792 申请日:2008-11-20
- 公开(公告)号:WO2009068214A3 公开(公告)日:2009-08-20
- 发明人: HEIMBACH DIRK , ROEHRIG SUSANNE , SCHNEIDER DIRK , RESTER ULRICH , BENDER ECKHARD , MEININGHAUS MARK , ZIMMERMANN KATJA , ZUBOV DIMITRY , BUCHMUELLER ANJA , DEGENFELD GEORGES , GERDES CHRISTOPH , GERISCH MICHAEL , GNOTH MARK JEAN , CANCHO-GRANDE YOLANDA , GERICKE KERSTEN MATTHIAS , JESKE MARIO
- 申请人: BAYER SCHERING PHARMA AG , HEIMBACH DIRK , ROEHRIG SUSANNE , SCHNEIDER DIRK , RESTER ULRICH , BENDER ECKHARD , MEININGHAUS MARK , ZIMMERMANN KATJA , ZUBOV DIMITRY , BUCHMUELLER ANJA , DEGENFELD GEORGES , GERDES CHRISTOPH , GERISCH MICHAEL , GNOTH MARK JEAN , CANCHO-GRANDE YOLANDA , GERICKE KERSTEN MATTHIAS , JESKE MARIO
- 专利权人: BAYER SCHERING PHARMA AG,HEIMBACH DIRK,ROEHRIG SUSANNE,SCHNEIDER DIRK,RESTER ULRICH,BENDER ECKHARD,MEININGHAUS MARK,ZIMMERMANN KATJA,ZUBOV DIMITRY,BUCHMUELLER ANJA,DEGENFELD GEORGES,GERDES CHRISTOPH,GERISCH MICHAEL,GNOTH MARK JEAN,CANCHO-GRANDE YOLANDA,GERICKE KERSTEN MATTHIAS,JESKE MARIO
- 当前专利权人: BAYER SCHERING PHARMA AG,HEIMBACH DIRK,ROEHRIG SUSANNE,SCHNEIDER DIRK,RESTER ULRICH,BENDER ECKHARD,MEININGHAUS MARK,ZIMMERMANN KATJA,ZUBOV DIMITRY,BUCHMUELLER ANJA,DEGENFELD GEORGES,GERDES CHRISTOPH,GERISCH MICHAEL,GNOTH MARK JEAN,CANCHO-GRANDE YOLANDA,GERICKE KERSTEN MATTHIAS,JESKE MARIO
- 优先权: DE102007057718 2007-11-30; DE102008010221 2008-02-20
- 主分类号: C07D413/04
- IPC分类号: C07D413/04 ; A61K31/454 ; A61K31/4545 ; A61P7/02 ; C07D413/14 ; C07D417/14
摘要:
The invention relates to novel heteroaryl-substituted piperidines, to a method for their production, to their use for the treatment and/or prophylaxis of diseases and to their use in the production of drugs for the treatment and/or prophylaxis of diseases, in particular cardiovascular diseases and tumours.
摘要(中):
本发明涉及新颖的杂芳基取代的哌啶,它们的制备方法,其用于疾病的治疗和/或预防和它们用于制备药物用于治疗和/或预防疾病用的使用,特别是心血管疾病和肿瘤性疾病的 ,
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D413/00 | 杂环化合物,含两个或更多个杂环,至少有1个环有氮原子和氧原子作为仅有的杂环原子 |
--------C07D413/02 | .含两个杂环 |
----------C07D413/04 | ..被环原子—环原子的键直接连接的 |