基本信息:
- 专利标题： BICYCLIC HETEROCYCLE DERIVATIVES AND METHODS OF USE THEREOF
- 专利标题（中）：双相异构体衍生物及其使用方法
- 申请号：PCT/US2008/080462 申请日：2008-10-20
- 公开(公告)号：WO2009055331A2 公开(公告)日：2009-04-30
- 发明人： XIA, Yan , BOYLE, Craig, D. , GREENLEE, William, J. , CHACKALAMANNIL, Samuel , JAYNE, Charles, Lee , STAMFORD, Andrew, W. , DAI, Xing , HARRIS, Joel, M. , NEUSTADT, Bernard, R. , NEELAMKAVIL, Santhosh, Francis , SHAH, Unmesh, G. , LANKIN, Claire, M. , LIU, Hong
- 申请人： SCHERING CORPORATION , XIA, Yan , BOYLE, Craig, D. , GREENLEE, William, J. , CHACKALAMANNIL, Samuel , JAYNE, Charles, Lee , STAMFORD, Andrew, W. , DAI, Xing , HARRIS, Joel, M. , NEUSTADT, Bernard, R. , NEELAMKAVIL, Santhosh, Francis , SHAH, Unmesh, G. , LANKIN, Claire, M. , LIU, Hong
- 申请人地址： 2000 Galloping Hill Road Kenilworth, New Jersey 07033-0530 US
- 专利权人： SCHERING CORPORATION,XIA, Yan,BOYLE, Craig, D.,GREENLEE, William, J.,CHACKALAMANNIL, Samuel,JAYNE, Charles, Lee,STAMFORD, Andrew, W.,DAI, Xing,HARRIS, Joel, M.,NEUSTADT, Bernard, R.,NEELAMKAVIL, Santhosh, Francis,SHAH, Unmesh, G.,LANKIN, Claire, M.,LIU, Hong
- 当前专利权人： SCHERING CORPORATION,XIA, Yan,BOYLE, Craig, D.,GREENLEE, William, J.,CHACKALAMANNIL, Samuel,JAYNE, Charles, Lee,STAMFORD, Andrew, W.,DAI, Xing,HARRIS, Joel, M.,NEUSTADT, Bernard, R.,NEELAMKAVIL, Santhosh, Francis,SHAH, Unmesh, G.,LANKIN, Claire, M.,LIU, Hong
- 当前专利权人地址： 2000 Galloping Hill Road Kenilworth, New Jersey 07033-0530 US
- 代理机构： BERGMAN, Jeffrey, P.
- 优先权： US60/981,677 20071022
- 主分类号： C07D451/06
- IPC分类号： C07D451/06 ; C07D471/08 ; C07D498/08 ; C07D487/08 ; C07D491/08 ; A61K31/46 ; A61K31/439 ; A61K31/506 ; A61K31/537 ; A61P3/00 ; C07D401/14 ; C07D495/08
摘要：
The present invention relates to Bicyclic Heterocycle Derivatives, compositions comprising a Bicyclic Heterocycle Derivative, and methods of using the Bicyclic Heterocycle Derivatives for treating or preventing obesity, diabetes, a metabolic disorder, a cardiovascular disease or a disorder related to the activity of GPR119 in a patient.
摘要（中）：
本发明涉及双环杂环衍生物，包含双环杂环衍生物的组合物，以及使用双环杂环衍生物治疗或预防肥胖症，糖尿病，代谢紊乱，心血管疾病或与GPR119活性相关的病症的方法 患者。
IPC结构图谱:
| C | 化学；冶金 |
| --C07 | 有机化学 |
| ----C07D | 杂环化合物 |
| ------C07D451/00 | 杂环化合物，含有8-氮杂二环 |
| --------C07D451/02 | .含有不进一步稠合的8-氮杂二环 |
| ----------C07D451/04 | ..有杂原子直接连在8-氮杂二环 |
| ------------C07D451/06 | ...氧原子 |