发明申请
WO2009016498A8 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS
审中-公开
基本信息:
- 专利标题： PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS
- 专利标题（中）：吡嗪和吡啶衍生物及其药物用途和组合物
- 申请号：PCT/IB2008002046 申请日：2008-07-29
- 公开(公告)号：WO2009016498A8 公开(公告)日：2010-11-11
- 发明人： SCHNUTE MARK E , CARROLL JEFFERY NEAL , HANAU CATHLEEN ELIZABETH , MCREYNOLDS MATTHEW DAVID , SCHOLTEN JEFFREY ALLEN , MCDONALD JOSEPH J , GRAPPERHAUS MARGARET L , MASSA MARK ALAN , RUMINSKI PETER G , SCHMIDT MICHELLE ANN , STROHBACH JOSEPH WALTER , HAMPER BRUCE CAMERON , FLETCHER THERESA R , ROGERS MICHAEL DAVID , O'BRIEN PATRICK MICHAEL , NAHRA JOE , MORRIS MARK ANTHONY , ROARK WILLIAM HOWARD
- 申请人： PFIZER , SCHNUTE MARK E , CARROLL JEFFERY NEAL , HANAU CATHLEEN ELIZABETH , MCREYNOLDS MATTHEW DAVID , SCHOLTEN JEFFREY ALLEN , MCDONALD JOSEPH J , GRAPPERHAUS MARGARET L , MASSA MARK ALAN , RUMINSKI PETER G , SCHMIDT MICHELLE ANN , STROHBACH JOSEPH WALTER , HAMPER BRUCE CAMERON , FLETCHER THERESA R , ROGERS MICHAEL DAVID , O'BRIEN PATRICK MICHAEL , NAHRA JOE , MORRIS MARK ANTHONY , ROARK WILLIAM HOWARD
- 专利权人： PFIZER,SCHNUTE MARK E,CARROLL JEFFERY NEAL,HANAU CATHLEEN ELIZABETH,MCREYNOLDS MATTHEW DAVID,SCHOLTEN JEFFREY ALLEN,MCDONALD JOSEPH J,GRAPPERHAUS MARGARET L,MASSA MARK ALAN,RUMINSKI PETER G,SCHMIDT MICHELLE ANN,STROHBACH JOSEPH WALTER,HAMPER BRUCE CAMERON,FLETCHER THERESA R,ROGERS MICHAEL DAVID,O'BRIEN PATRICK MICHAEL,NAHRA JOE,MORRIS MARK ANTHONY,ROARK WILLIAM HOWARD
- 当前专利权人： PFIZER,SCHNUTE MARK E,CARROLL JEFFERY NEAL,HANAU CATHLEEN ELIZABETH,MCREYNOLDS MATTHEW DAVID,SCHOLTEN JEFFREY ALLEN,MCDONALD JOSEPH J,GRAPPERHAUS MARGARET L,MASSA MARK ALAN,RUMINSKI PETER G,SCHMIDT MICHELLE ANN,STROHBACH JOSEPH WALTER,HAMPER BRUCE CAMERON,FLETCHER THERESA R,ROGERS MICHAEL DAVID,O'BRIEN PATRICK MICHAEL,NAHRA JOE,MORRIS MARK ANTHONY,ROARK WILLIAM HOWARD
- 优先权： US95360407 2007-08-02; US1553307 2007-12-20
- 主分类号： C07D401/04
- IPC分类号： C07D401/04 ; A61K31/44 ; A61K31/506 ; A61P19/00 ; A61P35/00 ; C07D401/14 ; C07D403/04 ; C07D405/04 ; C07D405/14 ; C07D413/14
摘要：
The prsent invention relates to compounds of Formula (I) and pharmaceutically acceptable salts thereof, processes for the preparation of, intermediates used in the preparation of, and compositions containing such compounds and the uses of such compounds as anti-inflammatory agents.
摘要（中）：
本发明涉及式（I）的化合物及其药学上可接受的盐，制备用途的中间体，含有这些化合物的组合物，以及这些化合物作为抗炎剂的用途。
IPC结构图谱:
| C | 化学；冶金 |
| --C07 | 有机化学 |
| ----C07D | 杂环化合物 |
| ------C07D401/00 | 杂环化合物，含有两个或更多个杂环，以氮原子作为仅有的杂环原子，至少有1个环是仅含有1个氮原子的六元环 |
| --------C07D401/02 | .含有两个杂环 |
| ----------C07D401/04 | ..被环原子—环原子的键直接连接的 |