发明申请
WO2008131859A3 USE OF CYCLICALLY SUBSTITUTED FUROPYRIMIDINE DERIVATIVES FOR TREATING PULMONARY ARTERIAL HYPERTONIA
审中-公开
基本信息:
- 专利标题: USE OF CYCLICALLY SUBSTITUTED FUROPYRIMIDINE DERIVATIVES FOR TREATING PULMONARY ARTERIAL HYPERTONIA
- 专利标题(中):VERWENDIMG环状的取代furopyrimidine衍生物对肺动脉高血压的治疗
- 申请号:PCT/EP2008003008 申请日:2008-04-16
- 公开(公告)号:WO2008131859A3 公开(公告)日:2009-07-16
- 发明人: LAMPE THOMAS , BECKER EVA-MARIA , KAST RAIMUND , BECK HARTMUT , JESKE MARIO , SCHUHMACHER JOACHIM , STOLL FRIEDERIKE , KLEIN MARTINA , AKBABA METIN , KNORR ANDREAS , STASCH JOHANNES-PETER , BAERFACKER LARS , HILLISCH ALEXANDER , KARIG GUNTER , MEININGHAUS MARK , SCHLEMMER KARL-HEINZ , SCHOHE-LOOP RUDOLF
- 申请人: BAYER SCHERING PHARMA AG , LAMPE THOMAS , BECKER EVA-MARIA , KAST RAIMUND , BECK HARTMUT , JESKE MARIO , SCHUHMACHER JOACHIM , STOLL FRIEDERIKE , KLEIN MARTINA , AKBABA METIN , KNORR ANDREAS , STASCH JOHANNES-PETER , BAERFACKER LARS , HILLISCH ALEXANDER , KARIG GUNTER , MEININGHAUS MARK , SCHLEMMER KARL-HEINZ , SCHOHE-LOOP RUDOLF
- 专利权人: BAYER SCHERING PHARMA AG,LAMPE THOMAS,BECKER EVA-MARIA,KAST RAIMUND,BECK HARTMUT,JESKE MARIO,SCHUHMACHER JOACHIM,STOLL FRIEDERIKE,KLEIN MARTINA,AKBABA METIN,KNORR ANDREAS,STASCH JOHANNES-PETER,BAERFACKER LARS,HILLISCH ALEXANDER,KARIG GUNTER,MEININGHAUS MARK,SCHLEMMER KARL-HEINZ,SCHOHE-LOOP RUDOLF
- 当前专利权人: BAYER SCHERING PHARMA AG,LAMPE THOMAS,BECKER EVA-MARIA,KAST RAIMUND,BECK HARTMUT,JESKE MARIO,SCHUHMACHER JOACHIM,STOLL FRIEDERIKE,KLEIN MARTINA,AKBABA METIN,KNORR ANDREAS,STASCH JOHANNES-PETER,BAERFACKER LARS,HILLISCH ALEXANDER,KARIG GUNTER,MEININGHAUS MARK,SCHLEMMER KARL-HEINZ,SCHOHE-LOOP RUDOLF
- 优先权: DE102007019690 2007-04-26
- 主分类号: A61K31/519
- IPC分类号: A61K31/519 ; A61P9/12 ; A61P11/00
摘要:
The invention relates to the use of cyclically substituted furopyrimidine derivatives of formula (I) for the treatment and/or prophylaxis of pulmonary arterial hypertonia and other forms of pulmonary hypertonia and to the use of said derivatives for producing medicaments for the treatment and/or prophylaxis of pulmonary arterial hypertonia and other forms of pulmonary hypertonia.
摘要(中):
本申请涉及使用式(I)为肺动脉高血压和其他形式的肺动脉高压以及它们用于制备药物用于治疗肺动脉高血压的治疗和/或预防中的用途在治疗和/或预防的环状取代furopyrimidine衍生物的 和其他形式的肺动脉高压。
IPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K31/00 | 含有机有效成分的医药配制品 |
--------A61K31/33 | .杂环化合物 |
----------A61K31/335 | ..仅有氧作为环杂原子的,例如制霉色基素 |
------------A61K31/40 | ...有仅以1个氮作为环杂原子的五元环的,例如舒必利、琥珀酰亚胺、托尔米丁、甲氧吡丁苯 |
--------------A61K31/50 | ....哒嗪;氢化哒嗪 |
----------------A61K31/519 | .....与杂环系统邻位或迫位稠合的 |