发明申请
WO2008117943A1 7-(3',4'-DIALKOXYPHENYL)-[1,2,4]-TRIAZOLO[1,5-A]PYRIMIDINE COMPOUNDS, PROCESS FOR PREPARING THEREOF, AND PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ARTHRITIS, ATOPIC DERMATITIS, TUMOR AND DEGENERATIVE BRAIN DISEASES COMPRISING THE SAME
审中-公开
基本信息:
- 专利标题: 7-(3',4'-DIALKOXYPHENYL)-[1,2,4]-TRIAZOLO[1,5-A]PYRIMIDINE COMPOUNDS, PROCESS FOR PREPARING THEREOF, AND PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ARTHRITIS, ATOPIC DERMATITIS, TUMOR AND DEGENERATIVE BRAIN DISEASES COMPRISING THE SAME
- 专利标题(中):7-(3',4'-二烷氧基苯基) - [1,2,4] - 三唑并[1,5-A]吡啶化合物,其制备方法和药物组合物,用于治疗或预防哮喘,慢性阻塞性肺动脉疾病, ARTHRITIS,ATOPIC DERMATITIS,TUMOR AND DEGE
- 申请号:PCT/KR2008/001278 申请日:2008-03-07
- 公开(公告)号:WO2008117943A1 公开(公告)日:2008-10-02
- 发明人: JEON, Dong Ju , NO, Zaesung , SONG, Jong Hwan , LEE, Gehyeong , KIM, Ikyon , PARK, Chang Min , CHEON, Hyae Gyeong , CHO, Young Sik , SONG, Jin Sook , BAE, Myung Ae , YOO, Sung-eun
- 申请人: KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY , JEON, Dong Ju , NO, Zaesung , SONG, Jong Hwan , LEE, Gehyeong , KIM, Ikyon , PARK, Chang Min , CHEON, Hyae Gyeong , CHO, Young Sik , SONG, Jin Sook , BAE, Myung Ae , YOO, Sung-eun
- 申请人地址: 100 Jang-dong, Yuseong-gu Daejeon 305-600 KR
- 专利权人: KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY,JEON, Dong Ju,NO, Zaesung,SONG, Jong Hwan,LEE, Gehyeong,KIM, Ikyon,PARK, Chang Min,CHEON, Hyae Gyeong,CHO, Young Sik,SONG, Jin Sook,BAE, Myung Ae,YOO, Sung-eun
- 当前专利权人: KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY,JEON, Dong Ju,NO, Zaesung,SONG, Jong Hwan,LEE, Gehyeong,KIM, Ikyon,PARK, Chang Min,CHEON, Hyae Gyeong,CHO, Young Sik,SONG, Jin Sook,BAE, Myung Ae,YOO, Sung-eun
- 当前专利权人地址: 100 Jang-dong, Yuseong-gu Daejeon 305-600 KR
- 代理机构: KWON, Oh-Sig et al.
- 优先权: KR10-2007-0028620 20070323
- 主分类号: C07D487/04
- IPC分类号: C07D487/04
摘要:
The present invention relates to novel {7-(3',4'-dialkoxyphenyl)-[1,2,4]-triazolo[1,5-a]pyrimidine compounds or pharmaceutically acceptable salts thereof, a process for preparing the same, and pharmaceutical compositions for treating or preventing inflammatory diseases including asthma and chronic obstructive pulmonary disease, arthritis, atopic dermatitis, cancers including leukemia, and degenerative brain diseases including Alzheimer's disease, depression and memory impairment, which comprises the same as an active ingredient.
摘要(中):
本发明涉及新的{7-(3',4'-二烷氧基苯基) - [1,2,4] - 三唑并[1,5-a]嘧啶化合物或其药学上可接受的盐,其制备方法, 以及用于治疗或预防包括哮喘和慢性阻塞性肺病,关节炎,特应性皮炎,包括白血病,包括阿尔茨海默氏病,抑郁症和记忆障碍在内的退行性脑疾病的炎症性疾病的药物组合物,其包含与活性成分相同的药物组合物。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D487/00 | 在稠环系中含有氮原子作为仅有的杂环原子的杂环化合物,不包含在C07D451/00至C07D477/00组中 |
--------C07D487/02 | .在稠合系中含有两个杂环 |
----------C07D487/04 | ..邻位稠合系 |