基本信息:
- 专利标题: PIPERIDINONES USEFUL IN THE TREATMENT OF INFLAMMATION
- 专利标题(中):哌啶酮可用于治疗炎症
- 申请号:PCT/GB2008/000854 申请日:2008-03-12
- 公开(公告)号:WO2008110793A1 公开(公告)日:2008-09-18
- 发明人: PELCMAN, Benjamin , KROG-JENSEN, Christian , SHEN, Yaping , YEE, James, Gee, Ken , MACKENZIE, Lloyd, F. , ZHOU, Yuanlin , HAN, Kang , RAYMOND, Jeffery, R.
- 申请人: BIOLIPOX AB , PELCMAN, Benjamin , KROG-JENSEN, Christian , SHEN, Yaping , YEE, James, Gee, Ken , MACKENZIE, Lloyd, F. , ZHOU, Yuanlin , HAN, Kang , RAYMOND, Jeffery, R.
- 申请人地址: Berzelius väg 3, plan 5 S-171 65 Solna SE
- 专利权人: BIOLIPOX AB,PELCMAN, Benjamin,KROG-JENSEN, Christian,SHEN, Yaping,YEE, James, Gee, Ken,MACKENZIE, Lloyd, F.,ZHOU, Yuanlin,HAN, Kang,RAYMOND, Jeffery, R.
- 当前专利权人: BIOLIPOX AB,PELCMAN, Benjamin,KROG-JENSEN, Christian,SHEN, Yaping,YEE, James, Gee, Ken,MACKENZIE, Lloyd, F.,ZHOU, Yuanlin,HAN, Kang,RAYMOND, Jeffery, R.
- 当前专利权人地址: Berzelius väg 3, plan 5 S-171 65 Solna SE
- 代理机构: MCNEENEY, Stephen
- 优先权: US60/906,804 20070312; US60/943,520 20070612; GB0722769.7 20071121
- 主分类号: C07D211/22
- IPC分类号: C07D211/22 ; C07D401/06 ; C07D407/06 ; C07D409/06 ; A61K31/45 ; A61P29/00 ; A61P35/00
摘要:
There is provided compounds of formula (I): wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , m and n have meanings given in the description, and pharmaceutically acceptable derivatives thereof, which compounds are useful in the treatment of diseases and conditions associated with inflammation.
摘要(中):
提供式(I)化合物:其中R 1,R 2,R 3,R 4, R 5,R 6,R 7,m和n具有本说明书中给出的含义及其药学上可接受的衍生物,该化合物是 可用于治疗与炎症相关的疾病和病症。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D211/00 | 杂环化合物,含氢化吡啶环,不与其他环稠合 |
--------C07D211/04 | .只有氢或碳原子直接连在环氮原子上 |
----------C07D211/06 | ..环原子间或环原子与非环原子间无双键 |
------------C07D211/08 | ...有烃基或取代的烃基直接连在环碳原子上 |
--------------C07D211/10 | ....有仅含碳原子和氢原子的基直接连在环碳原子上 |
----------------C07D211/20 | .....有被以单键键合的氧原子或硫原子取代的烃基 |
------------------C07D211/22 | ......被氧原子 |