发明申请
WO2008064217A9 CRYSTAL FORMS OF 2-(3-FLUORO-4-HYDROXYPHENYL)-7-VINYL-1,3-BENZOXAZOL-5-OL AND PHARMACEUTICAL FORMULATIONS THEREOF
审中-公开
基本信息:
- 专利标题: CRYSTAL FORMS OF 2-(3-FLUORO-4-HYDROXYPHENYL)-7-VINYL-1,3-BENZOXAZOL-5-OL AND PHARMACEUTICAL FORMULATIONS THEREOF
- 专利标题(中):2-(3-氟-4-羟基苯基)-7-乙烯基-1,3-苯并噻唑-5-OL及其药物制剂的晶体形式
- 申请号:PCT/US2007085226 申请日:2007-11-20
- 公开(公告)号:WO2008064217A9 公开(公告)日:2008-08-21
- 发明人: KRISHNAN MAHESH K , GHORAB MOHAMED , CARSON ROLLAND W , HASAN SHAMIM , NAGI ARWINDER , TADAYON ABDOLSAMAD , IERA SILVIO , MIRMEHRABI MAHMOUD
- 申请人: WYETH CORP , KRISHNAN MAHESH K , GHORAB MOHAMED , CARSON ROLLAND W , HASAN SHAMIM , NAGI ARWINDER , TADAYON ABDOLSAMAD , IERA SILVIO , MIRMEHRABI MAHMOUD
- 专利权人: WYETH CORP,KRISHNAN MAHESH K,GHORAB MOHAMED,CARSON ROLLAND W,HASAN SHAMIM,NAGI ARWINDER,TADAYON ABDOLSAMAD,IERA SILVIO,MIRMEHRABI MAHMOUD
- 当前专利权人: WYETH CORP,KRISHNAN MAHESH K,GHORAB MOHAMED,CARSON ROLLAND W,HASAN SHAMIM,NAGI ARWINDER,TADAYON ABDOLSAMAD,IERA SILVIO,MIRMEHRABI MAHMOUD
- 优先权: US86041506 2006-11-21; US86031706 2006-11-21; US86031806 2006-11-21; US86035206 2006-11-21; US86024806 2006-11-21; US86026506 2006-11-21; US86025306 2006-11-21; US86024606 2006-11-21
- 主分类号: C07D263/57
- IPC分类号: C07D263/57 ; A61K31/423 ; A61P15/00
摘要:
The present invention is directed to crystal forms (Forms B, D, E, and F described herein) of 2-
摘要(中):
本发明涉及2-形式的晶形(本文所述的形式B,D,E和F)
公开/授权文献:
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D263/00 | 杂环化合物,含有1,3-唑环或氢化1,3-唑环 |
--------C07D263/02 | .不和其他环稠合 |
----------C07D263/54 | ..苯并唑;氢化苯并唑 |
------------C07D263/56 | ...仅有氢原子、烃基或取代烃基,直接连在位置2上 |
--------------C07D263/57 | ....芳基或取代的芳基 |