发明申请
WO2008055870A8 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE
审中-公开
基本信息:
- 专利标题: GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE
- 专利标题(中):葡糖酰基 - 取代的苄基 - 苯并腈衍生物,含有该化合物的药物,其制备用途和制备方法
- 申请号:PCT/EP2007061877 申请日:2007-11-05
- 公开(公告)号:WO2008055870A8 公开(公告)日:2008-12-24
- 发明人: HIMMELSBACH FRANK , ECKHARDT MATTHIAS , EICKELMANN PETER , THOMAS LEO
- 申请人: BOEHRINGER INGELHEIM INT , BOEHRINGER INGELHEIM PHARMA , HIMMELSBACH FRANK , ECKHARDT MATTHIAS , EICKELMANN PETER , THOMAS LEO
- 专利权人: BOEHRINGER INGELHEIM INT,BOEHRINGER INGELHEIM PHARMA,HIMMELSBACH FRANK,ECKHARDT MATTHIAS,EICKELMANN PETER,THOMAS LEO
- 当前专利权人: BOEHRINGER INGELHEIM INT,BOEHRINGER INGELHEIM PHARMA,HIMMELSBACH FRANK,ECKHARDT MATTHIAS,EICKELMANN PETER,THOMAS LEO
- 优先权: EP06123515 2006-11-06; EP07102828 2007-02-21; EP07109727 2007-06-06
- 主分类号: C07H7/04
- IPC分类号: C07H7/04 ; A61K31/70 ; C07D309/10
摘要:
Glucopyranosyl-substituted benzyl-benzonitrile derivatives of general formula (I) as defined according to claim 1, including the tautomers, the stereoisomers thereof, the mixtures thereof and the salts thereof. The compounds according to the invention are suitable for the treatment of metabolic disorders.
摘要(中):
根据权利要求1定义的通式(I)的吡喃葡萄糖基取代的苄基 - 苄腈衍生物,包括其互变异构体,立体异构体,其混合物及其盐。 根据本发明的化合物适合于治疗代谢紊乱。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07H | 糖类;及其衍生物;核苷;核苷酸;核酸 |
------C07H7/00 | 含有以碳—碳键连在糖化物基团上的非糖化物基团的化合物 |
--------C07H7/04 | .碳环基 |