基本信息:
- 专利标题: PHTHALAZINONE DERIVATIVE
- 专利标题(中):邻苯二酚衍生物
- 申请号:PCT/GB2007/003888 申请日:2007-10-15
- 公开(公告)号:WO2008047082A2 公开(公告)日:2008-04-24
- 发明人: MENEAR, Keith, Allan , OTTRIDGE, Anthony, Peter , LONDESBROUGH, Derek, John , HALLETT, Michael, Raymond , MULLHOLLAND, Keith, Raymond , PITTAM, John, David , LAFFAN, David, Dermot, Patrick , ASHWORTH, Ian, Woodward , JONES, Martin, Francis , CHERRYMAN, Janette, Helen
- 申请人: KUDOS PHARMACEUTICALS LIMITED , MENEAR, Keith, Allan , OTTRIDGE, Anthony, Peter , LONDESBROUGH, Derek, John , HALLETT, Michael, Raymond , MULLHOLLAND, Keith, Raymond , PITTAM, John, David , LAFFAN, David, Dermot, Patrick , ASHWORTH, Ian, Woodward , JONES, Martin, Francis , CHERRYMAN, Janette, Helen
- 申请人地址: 15 Stanhope Gate London Greater London W1K 1LN GB
- 专利权人: KUDOS PHARMACEUTICALS LIMITED,MENEAR, Keith, Allan,OTTRIDGE, Anthony, Peter,LONDESBROUGH, Derek, John,HALLETT, Michael, Raymond,MULLHOLLAND, Keith, Raymond,PITTAM, John, David,LAFFAN, David, Dermot, Patrick,ASHWORTH, Ian, Woodward,JONES, Martin, Francis,CHERRYMAN, Janette, Helen
- 当前专利权人: KUDOS PHARMACEUTICALS LIMITED,MENEAR, Keith, Allan,OTTRIDGE, Anthony, Peter,LONDESBROUGH, Derek, John,HALLETT, Michael, Raymond,MULLHOLLAND, Keith, Raymond,PITTAM, John, David,LAFFAN, David, Dermot, Patrick,ASHWORTH, Ian, Woodward,JONES, Martin, Francis,CHERRYMAN, Janette, Helen
- 当前专利权人地址: 15 Stanhope Gate London Greater London W1K 1LN GB
- 代理机构: WATSON, Robert et al.
- 优先权: US60/829,694 20061017
- 主分类号: C07D237/32
- IPC分类号: C07D237/32 ; A61K31/502 ; A61P35/00
摘要:
4-[3-(4-cyclopropanecarbonyl-piperazine-1-carbonyl)-4-fluoro-benzyl]-2H-phthalazin-1-one as crystalline Form A.
摘要(中):
4- [3-(4-环丙烷羰基 - 哌嗪-1-羰基)-4-氟 - 苄基] -2H-酞嗪-1-酮,为晶型A.
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D237/00 | 杂环化合物,含1,2-二嗪环或氢化1,2-二嗪环 |
--------C07D237/02 | .不与其他环稠合 |
----------C07D237/30 | ..酞嗪 |
------------C07D237/32 | ...有氧原子直接连在含氮环的碳原子上 |