发明申请
WO2007115077A2 BICYCLIC BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS
审中-公开
基本信息:
- 专利标题: BICYCLIC BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS
- 专利标题(中):双环苯并咪唑化合物及其作为代谢型谷氨酸受体增效剂的用途
- 申请号:PCT/US2007065469 申请日:2007-03-29
- 公开(公告)号:WO2007115077A2 公开(公告)日:2007-10-11
- 发明人: EGLE IAN , ISAAC METHVIN , URBANEK REBECCA , MCLAREN FRANCES M , WALSH SALLY B , STEELMAN GARY B , BROWN DEAN G , NUGIEL DAVID , CHEN DEBORAH W , SLASSI ABDELMALIK , MA FUPENG
- 申请人: ASTRAZENECA AB , NPS PHARMA INC , EGLE IAN , ISAAC METHVIN , URBANEK REBECCA , MCLAREN FRANCES M , WALSH SALLY B , STEELMAN GARY B , BROWN DEAN G , NUGIEL DAVID , CHEN DEBORAH W , SLASSI ABDELMALIK , MA FUPENG
- 专利权人: ASTRAZENECA AB,NPS PHARMA INC,EGLE IAN,ISAAC METHVIN,URBANEK REBECCA,MCLAREN FRANCES M,WALSH SALLY B,STEELMAN GARY B,BROWN DEAN G,NUGIEL DAVID,CHEN DEBORAH W,SLASSI ABDELMALIK,MA FUPENG
- 当前专利权人: ASTRAZENECA AB,NPS PHARMA INC,EGLE IAN,ISAAC METHVIN,URBANEK REBECCA,MCLAREN FRANCES M,WALSH SALLY B,STEELMAN GARY B,BROWN DEAN G,NUGIEL DAVID,CHEN DEBORAH W,SLASSI ABDELMALIK,MA FUPENG
- 优先权: US78763406 2006-03-31
摘要:
Compounds of Formula (I): Formula (I) wherein A, B, D, L, R 1 , R 2 , R 3 , R 4 , m, and n are as defined for Formula (I) in the description. The invention also relates to processes for the preparation of the compounds and to new intermediates employed in the preparation, pharmaceutical compositions containing the compounds, and to the use of the compounds in therapy.
摘要(中):
式(I)化合物:其中A,B,D,L,R 1,R 2,R 3,R 3,R 4, R 4,m和n如说明书中对式(I)所定义。 本发明还涉及制备该化合物的方法和制备中使用的新中间体,含有该化合物的药物组合物,以及该化合物在治疗中的用途。