基本信息:
- 专利标题: ANTIBACTERIAL AGENTS
- 专利标题(中):抗菌剂
- 申请号:PCT/IB2005/001986 申请日:2005-07-13
- 公开(公告)号:WO2006013409A1 公开(公告)日:2006-02-09
- 发明人: DAS, Biswajit , KATOCH, Rita , HAJARE, Atul, Kashinath , KAPKOTI, Gobind, Singh , BANDYOPADHYAY, Anish , VENKATARAMANAN, Ramadass , KUMAR, Rajesh , KURHADE, Santosh, Haribhau , RATHY, Sujata , CHAKRABARTI, Anjan , SURASE, Yogesh, Bahan , SALMAN, Mohammad , RATTAN, Ashok
- 申请人: RANBAXY LABORATORIES LIMITED , DAS, Biswajit , KATOCH, Rita , HAJARE, Atul, Kashinath , KAPKOTI, Gobind, Singh , BANDYOPADHYAY, Anish , VENKATARAMANAN, Ramadass , KUMAR, Rajesh , KURHADE, Santosh, Haribhau , RATHY, Sujata , CHAKRABARTI, Anjan , SURASE, Yogesh, Bahan , SALMAN, Mohammad , RATTAN, Ashok
- 申请人地址: Plot No. 90, Sector - 32, Gurgaon, Haryana 122 001 IN
- 专利权人: RANBAXY LABORATORIES LIMITED,DAS, Biswajit,KATOCH, Rita,HAJARE, Atul, Kashinath,KAPKOTI, Gobind, Singh,BANDYOPADHYAY, Anish,VENKATARAMANAN, Ramadass,KUMAR, Rajesh,KURHADE, Santosh, Haribhau,RATHY, Sujata,CHAKRABARTI, Anjan,SURASE, Yogesh, Bahan,SALMAN, Mohammad,RATTAN, Ashok
- 当前专利权人: RANBAXY LABORATORIES LIMITED,DAS, Biswajit,KATOCH, Rita,HAJARE, Atul, Kashinath,KAPKOTI, Gobind, Singh,BANDYOPADHYAY, Anish,VENKATARAMANAN, Ramadass,KUMAR, Rajesh,KURHADE, Santosh, Haribhau,RATHY, Sujata,CHAKRABARTI, Anjan,SURASE, Yogesh, Bahan,SALMAN, Mohammad,RATTAN, Ashok
- 当前专利权人地址: Plot No. 90, Sector - 32, Gurgaon, Haryana 122 001 IN
- 优先权: IN1399/DEL/2004 20040728; IN1390/DEL/2005 20050530
- 主分类号: C07H17/08
- IPC分类号: C07H17/08 ; A61K31/7048 ; A61P31/04
摘要:
The present invention provides acylide derivatives, which can be used as antibacterial agents. Compounds disclosed herein can be used for the treatment or prevention of a condition caused by or contributed to by Gram-positive, Gram-negative or anaerobic bacteria, more particularly against bacterium such as Staphylococci, Streptococci, Enterococci, Haemophilus, Moraxalla spp., Chlamydia spp., Mycoplasm, Legionella spp., My obacterium, Helicobacter, Clostridium, Bacteroides, Corynebacterium, B ccillus or Enterobactericeae. Processes for the preparation of disclosed compounds, pharmaceutical compositions thereof, and method of treating bacterial infections, are also provided.
摘要(中):
本发明提供可用作抗菌剂的酰化物衍生物。 本文公开的化合物可用于治疗或预防由革兰氏阳性,革兰氏阴性或厌氧细菌引起的或由其贡献的病症,特别是针对细菌如葡萄球菌,链球菌,肠球菌,嗜血杆菌,莫萨拉氏菌,衣原体 肉豆蔻,军团菌,我的杆菌,幽门螺杆菌,梭菌属,拟杆菌属,棒状杆菌属,B肠杆菌属或肠杆菌属。 还提供了制备所公开的化合物的方法,其药物组合物和治疗细菌感染的方法。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07H | 糖类;及其衍生物;核苷;核苷酸;核酸 |
------C07H17/00 | 含有直接连在糖化物基团的杂原子上的杂环基的化合物 |
--------C07H17/04 | .仅含有氧作为杂环原子的杂环基 |
----------C07H17/08 | ..含有八元或更多元的杂环,如红霉素 |