发明申请
WO2005066139A2 2-(AMINO-SUBSTITUTED)-4-ARYL PYRAMIDINES AND RELATED COMPOUNDS USEFUL FOR TREATING INFLAMMATORY DISEASES
审中-公开
基本信息:
- 专利标题: 2-(AMINO-SUBSTITUTED)-4-ARYL PYRAMIDINES AND RELATED COMPOUNDS USEFUL FOR TREATING INFLAMMATORY DISEASES
- 专利标题(中):2-氨基取代的4-亚氨基吡啶和相关化合物用于治疗炎症性疾病
- 申请号:PCT/US2005/000663 申请日:2005-01-10
- 公开(公告)号:WO2005066139A2 公开(公告)日:2005-07-21
- 发明人: FLEMING, Paul, E. , SHI, Zhan , CHEN, Shaowu , SCHMIDT, Jane, F. , READER, John, C. , HONE, Neal, D. , CIAVARRI, Jefrey, P.
- 申请人: MILLENNIUM PHARMACEUTICALS, INC. , FLEMING, Paul, E. , SHI, Zhan , CHEN, Shaowu , SCHMIDT, Jane, F. , READER, John, C. , HONE, Neal, D. , CIAVARRI, Jefrey, P.
- 申请人地址: 40 Landsdowne Street, Cambridge, MA 02139 US
- 专利权人: MILLENNIUM PHARMACEUTICALS, INC.,FLEMING, Paul, E.,SHI, Zhan,CHEN, Shaowu,SCHMIDT, Jane, F.,READER, John, C.,HONE, Neal, D.,CIAVARRI, Jefrey, P.
- 当前专利权人: MILLENNIUM PHARMACEUTICALS, INC.,FLEMING, Paul, E.,SHI, Zhan,CHEN, Shaowu,SCHMIDT, Jane, F.,READER, John, C.,HONE, Neal, D.,CIAVARRI, Jefrey, P.
- 当前专利权人地址: 40 Landsdowne Street, Cambridge, MA 02139 US
- 代理机构: SHAIR, Karoline, K., M.
- 优先权: US60/534.898 20040108
- 主分类号: C07D239/00
- IPC分类号: C07D239/00
摘要:
A heterocyclic inhibitor having the formula (I), with the variables defined herein, which is useful for treating inflammatory and other physiological disorders in which PKC-theta isoform plays a role.
摘要(中):
具有式(I)的杂环抑制剂,具有本文定义的变量,其可用于治疗其中PKC-θ同种型起作用的炎性和其他生理障碍。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D239/00 | 杂环化合物,含1,3-二嗪环或氢化1,3-二嗪环 |