基本信息:
- 专利标题: AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS
- 专利标题(中):作为CANNABINOID受体调节剂的偶氮异构体
- 申请号:PCT/US2004/042878 申请日:2004-12-17
- 公开(公告)号:WO2005063762A1 公开(公告)日:2005-07-14
- 发明人: GU, Guixue , EWING, William, R. , MIKKILINENI, Amarendra, B. , PENDRI, Annapurna , ELLSWORTH, Bruce, A. , SHER, Philip, M. , GERRITZ, Samuel , SUN, Chongqing , MURUGESAN, Natesan , WU, Ximao
- 申请人: BRISTOL-MYERS SQUIBB COMPANY , GU, Guixue , EWING, William, R. , MIKKILINENI, Amarendra, B. , PENDRI, Annapurna , ELLSWORTH, Bruce, A. , SHER, Philip, M. , GERRITZ, Samuel , SUN, Chongqing , MURUGESAN, Natesan , WU, Ximao
- 申请人地址: Route 206 and Province Line Road, Princeton, New Jersey 08543-4000 US
- 专利权人: BRISTOL-MYERS SQUIBB COMPANY,GU, Guixue,EWING, William, R.,MIKKILINENI, Amarendra, B.,PENDRI, Annapurna,ELLSWORTH, Bruce, A.,SHER, Philip, M.,GERRITZ, Samuel,SUN, Chongqing,MURUGESAN, Natesan,WU, Ximao
- 当前专利权人: BRISTOL-MYERS SQUIBB COMPANY,GU, Guixue,EWING, William, R.,MIKKILINENI, Amarendra, B.,PENDRI, Annapurna,ELLSWORTH, Bruce, A.,SHER, Philip, M.,GERRITZ, Samuel,SUN, Chongqing,MURUGESAN, Natesan,WU, Ximao
- 当前专利权人地址: Route 206 and Province Line Road, Princeton, New Jersey 08543-4000 US
- 代理机构: DUNCAN, Sammy, G., Jr.
- 优先权: US60/531,451 20031219; US11/016,198 20041217
- 主分类号: C07D487/04
- IPC分类号: C07D487/04
摘要:
The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and optionally one or more additional therapeutic agents and methods of treatment using the compounds according to Formula I both alone and in combination with one or more additional therapeutic agents. The compounds have the general Formula I. including all prodrugs, pharmaceutically acceptable salts and stereoisomers, R 1 , R 2 , R 3 , R 4 , R 5 , m and n are described herein.
摘要(中):
本申请描述了根据式I的化合物,包含至少一种根据式I的化合物和任选的一种或多种另外的治疗剂的药物组合物和使用根据式I的化合物的治疗方法,其单独和与一种或多种另外的 治疗剂。 该化合物具有通式I.包括所有前药,药学上可接受的盐和立体异构体,R 1,R 2,R 3,R 4,R 5,m和n如本文所述。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D487/00 | 在稠环系中含有氮原子作为仅有的杂环原子的杂环化合物,不包含在C07D451/00至C07D477/00组中 |
--------C07D487/02 | .在稠合系中含有两个杂环 |
----------C07D487/04 | ..邻位稠合系 |