基本信息:
- 专利标题: THERAPEUTIC PHOSPHONATE COMPOUNDS
- 申请号:PCT/US2004/013283 申请日:2004-04-26
- 公开(公告)号:WO2005002626A2 公开(公告)日:2005-01-13
- 发明人: BOOJAMRA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , DESAI, Manoj , FARDIS, Maria , GIBBS, Craig, S. , HIRSCHMANN, Ralph, F. , HUANG, Alan, X. , JIN, Haolun , KIM, Choung, U. , KIRSCHBERG, Thorsten, A. , KRAWCZYK, Steven , LEE, Christopher, P. , LEE, William, A. , LIN, Kuei-Ying , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , NELSON, Peter, H. , OARE, David, A. , PRASAD, Vidya, K. , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, William, J. , ZHANG, Jennifer, R. , ZHANG, Lijun
- 申请人: GILEAD SCIENCES, INC. , BOOJAMRA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , DESAI, Manoj , FARDIS, Maria , GIBBS, Craig, S. , HIRSCHMANN, Ralph, F. , HUANG, Alan, X. , JIN, Haolun , KIM, Choung, U. , KIRSCHBERG, Thorsten, A. , KRAWCZYK, Steven , LEE, Christopher, P. , LEE, William, A. , LIN, Kuei-Ying , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , NELSON, Peter, H. , OARE, David, A. , PRASAD, Vidya, K. , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, William, J. , ZHANG, Jennifer, R. , ZHANG, Lijun
- 申请人地址: 333 Lakeside Drive, Foster City, CA 94404 US
- 专利权人: GILEAD SCIENCES, INC.,BOOJAMRA, Constantine, G.,CANNIZZARO, Carina, E.,CHEN, James, M.,CHEN, Xiaowu,CHO, Aesop,CHONG, Lee, S.,DESAI, Manoj,FARDIS, Maria,GIBBS, Craig, S.,HIRSCHMANN, Ralph, F.,HUANG, Alan, X.,JIN, Haolun,KIM, Choung, U.,KIRSCHBERG, Thorsten, A.,KRAWCZYK, Steven,LEE, Christopher, P.,LEE, William, A.,LIN, Kuei-Ying,MACKMAN, Richard, L.,MARKEVITCH, David, Y.,NELSON, Peter, H.,OARE, David, A.,PRASAD, Vidya, K.,PYUN, Hyung-Jung,RAY, Adrian, S.,SHERLOCK, Rosemarie,SWAMINATHAN, Sundaramoorthi,WATKINS, William, J.,ZHANG, Jennifer, R.,ZHANG, Lijun
- 当前专利权人: GILEAD SCIENCES, INC.,BOOJAMRA, Constantine, G.,CANNIZZARO, Carina, E.,CHEN, James, M.,CHEN, Xiaowu,CHO, Aesop,CHONG, Lee, S.,DESAI, Manoj,FARDIS, Maria,GIBBS, Craig, S.,HIRSCHMANN, Ralph, F.,HUANG, Alan, X.,JIN, Haolun,KIM, Choung, U.,KIRSCHBERG, Thorsten, A.,KRAWCZYK, Steven,LEE, Christopher, P.,LEE, William, A.,LIN, Kuei-Ying,MACKMAN, Richard, L.,MARKEVITCH, David, Y.,NELSON, Peter, H.,OARE, David, A.,PRASAD, Vidya, K.,PYUN, Hyung-Jung,RAY, Adrian, S.,SHERLOCK, Rosemarie,SWAMINATHAN, Sundaramoorthi,WATKINS, William, J.,ZHANG, Jennifer, R.,ZHANG, Lijun
- 当前专利权人地址: 333 Lakeside Drive, Foster City, CA 94404 US
- 代理机构: BOSSE, Mark, L.
- 优先权: US60/465,594 20030425; US60/465,630 20030425; US60/465,400 20030425; US60/465,639 20030425; US60/465,602 20030425; US60/465,587 20030425; US60/465,463 20030425; US60/465,728 20030425; US60/465,601 20030425; US60/465,550 20030425; US60/465,633 20030425; US60/465,598 20030425; US60/465,473 20030425; US60/465,472 20030425; US60/465,546 20030425; US60/465,593 20030425; US60/465,667 20030425; US60/465,698 20030425; US60/465,537 20030425; US60/465,634 20030425; US60/465,720 20030425; US60/465,600 20030425; US60/465,347 20030425; US60/465,469 20030425; US60/465,690 20030425; US60/465,649 20030425; US60/465,742 20030425; US60/465,647 20030425; US60/465,821 20030425; US60/465,591 20030425; US60/465,548 20030425; US60/465,561 20030425; US60/465,553 20030425; US60/465,554 20030425; US60/465,684 20030425; US60/465,478 20030425; US60/465,289 20030425; US60/465,588 20030425; US60/465,759 20030425; US60/465,687 20030425; US60/465,584 20030425; US60/465,610 20030425; US60/465,589 20030425; US60/465,714 20030425; US60/465,631 20030425; US60/465,559 20030425; US60/465,467 20030425; US60/465,569 20030425; US60/465,465 20030425; US60/465,545 20030425; US60/465,567 20030425; US60/465,471 20030425; US60/465,343 20030425; US60/465,287 20030425; US60/465,668 20030425; US60/465,452 20030425; US60/465,620 20030425; US60/465,682 20030425; US60/465,683 20030425; US60/465,614 20030425; US60/465,641 20030425; US60/465,603 20030425; US60/465,394 20030425; US60/465,536 20030425; US60/465,406 20030425; US60/465,746 20030425; US60/465,695 20030425; US60/465,547 20030425; US60/465,335 20030425; US60/465,449 20030425; US60/465,696 20030425; US60/465,408 20030425; US60/465,608 20030425; US60/465,586 20030425; US60/465,607 20030425; US60/465,479 20030425; US60/465,640 20030425; US60/465,632 20030425; US60/465,342 20030425; US60/465,422 20030425; US60/465,560 20030425; US60/465,332 20030425; US60/465,638 20030425; US60/465,749 20030425; US60/465,480 20030425; US60/495,757 20030814; US60/495,687 20030815; US60/495,298 20030815; US60/495,805 20030815; US60/495,684 20030815; US60/495,490 20030815; US60/495,600 20030815; US60/495,487 20030815; US60/495,390 20030815; US60/495,342 20030815; US60/495,391 20030815; US60/495,564 20030815; US60/495,492 20030815; US60/495,772 20030815; US60/495,964 20030815; US60/495,317 20030815; US60/495,491 20030815; US60/495,453 20030815; US60/495,760 20030815; US60/495,592 20030815; US60/495,763 20030815; US60/495,345 20030815; US60/495,273 20030815; US60/495,602 20030815; US60/495,343 20030815; US60/495,275 20030815; US60/495,630 20030815; US60/495,277 20030815; US60/495,485 20030815; US60/495,278 20030815; US60/495,430 20030815; US60/495,344 20030815; US60/495,334 20030815; US60/495,671 20030815; US60/495,696 20030815; US60/495,349 20030815; US60/495,633 20030815; US60/495,632 20030815; US60/495,631 20030815; US60/495,539 20030815; US60/495,341 20030815; US60/495,382 20030815; US60/495,388 20030815; US60/495,525 20030815; US60/495,387 20030815; US60/495,686 20030815; US60/495,629 20030815; US60/495,527 20030815; US60/495,685 20030815; US60/495,484 20030815; US60/495,644 20030815; US60/495,297 20030815; US60/495,682 20030815; US60/513,564 20031024; US60/513,588 20031024
- 主分类号: A61K47/48
- IPC分类号: A61K47/48
摘要:
The invention is related to phosphorus substituted therapeutic agents, compositions containing such phosphorus substituted agents, and therapeutic methods that include the administration of such phosphorus substituted agents, as well as to processes and intermediates useful for preparing such agents.
公开/授权文献:
- WO2005002626A3 THERAPEUTIC PHOSPHONATE COMPOUNDS 公开/授权日:2005-01-13
IPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K47/00 | 以所用的非有效成分为特征的医用配制品,如载体、惰性添加剂 |
--------A61K47/48 | .非有效成分被化学键键合到有效成分上,例如聚合物药物轭合物 |