基本信息:
- 专利标题: PROTON-SENSING G-PROTEIN COUPLED RECEPTORS AND DNA SEQUENCES THEREOF
- 专利标题(中):丙型肝炎病毒感染G蛋白偶联受体及其DNA序列
- 申请号:PCT/EP2004/006625 申请日:2004-06-18
- 公开(公告)号:WO2004112823A1 公开(公告)日:2004-12-29
- 发明人: BAUMGARTEN, Birgit , JONES, Carol, Elizabeth , LUDWIG, Marie-Gabrielle , MARTINY-BARON, Georg , SEUWEN, Klaus , WOLF, Romain , WYDER, Lorenza , SUPLY, Thomas
- 申请人: NOVARTIS AG , NOVARTIS PHARMA GMBH , BAUMGARTEN, Birgit , JONES, Carol, Elizabeth , LUDWIG, Marie-Gabrielle , MARTINY-BARON, Georg , SEUWEN, Klaus , WOLF, Romain , WYDER, Lorenza , SUPLY, Thomas
- 申请人地址: Lichtstrasse 35, CH-4056 Basel CH
- 专利权人: NOVARTIS AG,NOVARTIS PHARMA GMBH,BAUMGARTEN, Birgit,JONES, Carol, Elizabeth,LUDWIG, Marie-Gabrielle,MARTINY-BARON, Georg,SEUWEN, Klaus,WOLF, Romain,WYDER, Lorenza,SUPLY, Thomas
- 当前专利权人: NOVARTIS AG,NOVARTIS PHARMA GMBH,BAUMGARTEN, Birgit,JONES, Carol, Elizabeth,LUDWIG, Marie-Gabrielle,MARTINY-BARON, Georg,SEUWEN, Klaus,WOLF, Romain,WYDER, Lorenza,SUPLY, Thomas
- 当前专利权人地址: Lichtstrasse 35, CH-4056 Basel CH
- 代理机构: GRUBB, Philipp
- 优先权: US60/480,245 200306020; US60/499,549 20030902
- 主分类号: A61K38/17
- IPC分类号: A61K38/17
摘要:
This invention relates to the newly identified utility of certain G protein-coupled receptors (GPCRs), in particular to OGR1, GPR4 and TDAG8 (TDAG8 is also named GPR65) polypeptides, and polynucleotides encoding such GPCR polypeptides, to their use in diagnosis and to methods of identifying compounds that are agonists or antagonists to said GPCRs, and to the production of such polypeptides and polynucleotides.
摘要(中):
本发明涉及新鉴定的某些G蛋白偶联受体(GPCR),特别是OGR1,GPR4和TDAG8(TDAG8也称为GPR65)多肽以及编码这种GPCR多肽的多核苷酸在临床诊断中的用途和 识别作为所述GPCR的激动剂或拮抗剂的化合物的方法,以及这些多肽和多核苷酸的产生。
IPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K38/00 | 含肽的医药配制品 |
--------A61K38/04 | .在完全确定的序列中最多有20个氨基酸的肽;其衍生物 |
----------A61K38/17 | ..来源于动物;来源于人类 |