基本信息:
- 专利标题: DIPEPTIDYL PEPTIDASE INHIBITORS
- 专利标题(中):DIPEPTIDYL PEPTIDASE抑制剂
- 申请号:PCT/US2004/015211 申请日:2004-05-13
- 公开(公告)号:WO2004103993A1 公开(公告)日:2004-12-02
- 发明人: FENG, Jun , GWALTNEY, Stephen L. , STAFFORD, Jeffrey A. , WALLACE, Michael B. , XIAO, Xiao-Yi , ZHANG, Zhiyuan
- 申请人: SYRRX, INC. , FENG, Jun , GWALTNEY, Stephen L. , STAFFORD, Jeffrey A. , WALLACE, Michael B. , XIAO, Xiao-Yi , ZHANG, Zhiyuan
- 申请人地址: 10410 Science Center Drive, San Diego, California 92121 US
- 专利权人: SYRRX, INC.,FENG, Jun,GWALTNEY, Stephen L.,STAFFORD, Jeffrey A.,WALLACE, Michael B.,XIAO, Xiao-Yi,ZHANG, Zhiyuan
- 当前专利权人: SYRRX, INC.,FENG, Jun,GWALTNEY, Stephen L.,STAFFORD, Jeffrey A.,WALLACE, Michael B.,XIAO, Xiao-Yi,ZHANG, Zhiyuan
- 当前专利权人地址: 10410 Science Center Drive, San Diego, California 92121 US
- 代理机构: WEITZ, David J.
- 优先权: US60/470,523 20030514
- 主分类号: C07D403/12
- IPC分类号: C07D403/12
摘要:
Pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound with the formula: (I) where the labeled substituents are as described herein.
摘要(中):
提供药物,试剂盒和方法用于DPP-IV和其它S9蛋白酶,其包含具有下式的化合物:(I)其中标记的取代基如本文所述。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D403/00 | 杂环化合物,含有两个或更多的杂环,以氮原子作为仅有的杂环原子,C07D401/00组不包含的 |
--------C07D403/02 | .含两个杂环 |
----------C07D403/12 | ..被含有杂原子的链作为键链连接的 |