发明申请
WO2004101508A3 SYNTHETIC TECHNIQUES AND INTERMEDIATES FOR POLYHYDROXY DIENYL LACTONES AND MIMICS THEREOF
审中-公开
基本信息:
- 专利标题: SYNTHETIC TECHNIQUES AND INTERMEDIATES FOR POLYHYDROXY DIENYL LACTONES AND MIMICS THEREOF
- 专利标题(中):聚羟基二烯丙基内酯及其模拟物的合成工艺及中间体
- 申请号:PCT/US2004010272 申请日:2004-04-02
- 公开(公告)号:WO2004101508A3 公开(公告)日:2005-03-03
- 发明人: MYLES DAVID C , BURLINGAME MARK , SHAW SIMON JAMES , SUNDERMANN KURT F , FREEZE BRIAN SCOTT , MARTIN IGNACIO BROUARD , HIROSE TOMOYASU , SMITH AMOS B
- 申请人: UNIV PENNSYLVANIA , MYLES DAVID C , BURLINGAME MARK , SHAW SIMON JAMES , SUNDERMANN KURT F , FREEZE BRIAN SCOTT , MARTIN IGNACIO BROUARD , HIROSE TOMOYASU , SMITH AMOS B
- 专利权人: UNIV PENNSYLVANIA,MYLES DAVID C,BURLINGAME MARK,SHAW SIMON JAMES,SUNDERMANN KURT F,FREEZE BRIAN SCOTT,MARTIN IGNACIO BROUARD,HIROSE TOMOYASU,SMITH AMOS B
- 当前专利权人: UNIV PENNSYLVANIA,MYLES DAVID C,BURLINGAME MARK,SHAW SIMON JAMES,SUNDERMANN KURT F,FREEZE BRIAN SCOTT,MARTIN IGNACIO BROUARD,HIROSE TOMOYASU,SMITH AMOS B
- 优先权: US46074403 2003-04-02; US47637803 2003-06-06
- 主分类号: C07D
- IPC分类号: C07D20060101 ; C07D309/10 ; C07D309/30 ; C07D309/32 ; C07F9/28
摘要:
Synthetic methods and intermediates useful in the preparation of lactone containing compounds such as discodermolide and compounds which mimic the chemical or biological activity of discodermolide are provided.
摘要(中):
提供了用于制备含内酯化合物如discodermolide的合成方法和中间体以及模拟discodermolide化学或生物活性的化合物。