基本信息:
- 专利标题: NEW FORMS OF CABERGOLINE
- 专利标题(中):新形态的碳酸氢钠
- 申请号:PCT/IB2004/002512 申请日:2004-04-20
- 公开(公告)号:WO2004094368A2 公开(公告)日:2004-11-04
- 发明人: GUTMAN, Arie , TISHIN, Boris , VILENSKI, Alex , AGAZADE, Albay , PERTZIKOV, Boris , NISNEVICH, Gennady
- 申请人: FINETECH LABORATORIES, LTD. , GUTMAN, Arie , TISHIN, Boris , VILENSKI, Alex , AGAZADE, Albay , PERTZIKOV, Boris , NISNEVICH, Gennady
- 申请人地址: Technion City, P.O. Box 3557, 31032 Haifa IL
- 专利权人: FINETECH LABORATORIES, LTD.,GUTMAN, Arie,TISHIN, Boris,VILENSKI, Alex,AGAZADE, Albay,PERTZIKOV, Boris,NISNEVICH, Gennady
- 当前专利权人: FINETECH LABORATORIES, LTD.,GUTMAN, Arie,TISHIN, Boris,VILENSKI, Alex,AGAZADE, Albay,PERTZIKOV, Boris,NISNEVICH, Gennady
- 当前专利权人地址: Technion City, P.O. Box 3557, 31032 Haifa IL
- 优先权: IL155545 20030421
- 主分类号: C07D
- IPC分类号: C07D
摘要:
The invention provides methods for preparing amorphous physical form of cabergoline, and solvate form A of cabergoline useful in the preparation of the first mentioned physical form. A method for treating a prolactin disorder with medicaments prepared from amorphous physical form of cabergoline and solvate form A of cabergoline is also disclosed.
摘要(中):
本发明提供了制备卡麦角林的无定形物理形式的方法,以及用于制备第一种物理形式的卡麦角林的溶剂化物A. 还公开了用卡麦角林的无定形物理形式和卡麦角林的溶剂合物形式A制备的药物治疗催乳素障碍的方法。