发明申请
WO2004089911A1 PYRAZOLE DERIVATIVES AS GAMMA-SECRETASE INHIBITORS USEFUL IN THE TREATMENT OF ALZHEIMER’S DISEASE
审中-公开
基本信息:
- 专利标题: PYRAZOLE DERIVATIVES AS GAMMA-SECRETASE INHIBITORS USEFUL IN THE TREATMENT OF ALZHEIMER’S DISEASE
- 专利标题(中):用作治疗阿尔茨海默病的GAMMA-分泌酶抑制剂的吡唑衍生物
- 申请号:PCT/GB2004/001452 申请日:2004-04-01
- 公开(公告)号:WO2004089911A1 公开(公告)日:2004-10-21
- 发明人: BETTATI, Michela , CHAMBERS, Mark, Stuart , HUNT, Peter, Alan , JONES, Philip , MACLEOD, Angus, Murray , SZEKERES, Helen, Jane , TEALL, Martin, Richard
- 申请人: MERCK SHARP & DOHME LIMITED , BETTATI, Michela , CHAMBERS, Mark, Stuart , HUNT, Peter, Alan , JONES, Philip , MACLEOD, Angus, Murray , SZEKERES, Helen, Jane , TEALL, Martin, Richard
- 申请人地址: Hertford Road, Hoddesdon Hertfordshire EN11 9BU GB
- 专利权人: MERCK SHARP & DOHME LIMITED,BETTATI, Michela,CHAMBERS, Mark, Stuart,HUNT, Peter, Alan,JONES, Philip,MACLEOD, Angus, Murray,SZEKERES, Helen, Jane,TEALL, Martin, Richard
- 当前专利权人: MERCK SHARP & DOHME LIMITED,BETTATI, Michela,CHAMBERS, Mark, Stuart,HUNT, Peter, Alan,JONES, Philip,MACLEOD, Angus, Murray,SZEKERES, Helen, Jane,TEALL, Martin, Richard
- 当前专利权人地址: Hertford Road, Hoddesdon Hertfordshire EN11 9BU GB
- 代理机构: BUCHAN, Gavin, MacNicol
- 优先权: GB0308318.5 20030410
- 主分类号: C07D231/12
- IPC分类号: C07D231/12
摘要:
The compounds of formula (I): inhibit gamma-secretase and hence are of utility in the treatment or prevention of Alzheimer's disease.
摘要(中):
式(I)化合物:抑制γ-分泌酶,因此可用于治疗或预防阿尔茨海默氏病。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D231/00 | 杂环化合物,含1,2-二唑或氢化1,2-二唑环 |
--------C07D231/02 | .不与其他环稠合 |
----------C07D231/06 | ..环原子间或环原子与非环原子间有1个双键 |
------------C07D231/12 | ...只有氢原子、烃基或取代的烃基,直接连在环碳原子上 |