发明申请
WO2004011446A1 INDANE, DIHYDROBENZOFURAN, AND TETRAHYDRONAPHTHALENE CARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ANTIDIABETICS
审中-公开
基本信息:
- 专利标题: INDANE, DIHYDROBENZOFURAN, AND TETRAHYDRONAPHTHALENE CARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ANTIDIABETICS
- 专利标题(中):吲哚,二氢苯并呋喃和四氢萘基羧酸衍生物及其作为抗生素的用途
- 申请号:PCT/US2003/023342 申请日:2003-07-25
- 公开(公告)号:WO2004011446A1 公开(公告)日:2004-02-05
- 发明人: WICKENS, Philip , CANTIN, Louis-David , CHUANG, Chih-Yuan , DAI, Miao , HENTEMANN, Martin, F. , KUMARASINGHE, Ellalahewage , LIANG, Sidney, X. , LOWE, Derek, B. , SHELEKHIN, Tatiana, E. , WANG, Yamin , ZHANG, Chengzhi , ZHANG, Hai-Jun , ZHAO, Qian
- 申请人: BAYER PHARMACEUTICALS CORPORATION , WICKENS, Philip , CANTIN, Louis-David , CHUANG, Chih-Yuan , DAI, Miao , HENTEMANN, Martin, F. , KUMARASINGHE, Ellalahewage , LIANG, Sidney, X. , LOWE, Derek, B. , SHELEKHIN, Tatiana, E. , WANG, Yamin , ZHANG, Chengzhi , ZHANG, Hai-Jun , ZHAO, Qian
- 申请人地址: 400 Morgan Lane, West Haven, CT 06516 US
- 专利权人: BAYER PHARMACEUTICALS CORPORATION,WICKENS, Philip,CANTIN, Louis-David,CHUANG, Chih-Yuan,DAI, Miao,HENTEMANN, Martin, F.,KUMARASINGHE, Ellalahewage,LIANG, Sidney, X.,LOWE, Derek, B.,SHELEKHIN, Tatiana, E.,WANG, Yamin,ZHANG, Chengzhi,ZHANG, Hai-Jun,ZHAO, Qian
- 当前专利权人: BAYER PHARMACEUTICALS CORPORATION,WICKENS, Philip,CANTIN, Louis-David,CHUANG, Chih-Yuan,DAI, Miao,HENTEMANN, Martin, F.,KUMARASINGHE, Ellalahewage,LIANG, Sidney, X.,LOWE, Derek, B.,SHELEKHIN, Tatiana, E.,WANG, Yamin,ZHANG, Chengzhi,ZHANG, Hai-Jun,ZHAO, Qian
- 当前专利权人地址: 400 Morgan Lane, West Haven, CT 06516 US
- 代理机构: GREENMAN, Jeffrey, M.
- 优先权: US60/399,095 20020726
- 主分类号: C07D263/32
- IPC分类号: C07D263/32
摘要:
This invention relates to novel indane, dihydrobenzofuran, and tetrahydronaphthalene carboxylic acid derivatives whice are useful in the treatment of diseases such sa diabetes, diabetes-related disorders, obesity, hyperlipidemia, and cardiovascular diseases. The invention also relates to intermediates useful in preparation of said carboxylic derivatives and to methods of preparation.
摘要(中):
本发明涉及新颖的茚满二氢苯并呋喃和四氢萘羧酸衍生物,其可用于治疗诸如糖尿病,糖尿病相关疾病,肥胖症,高脂血症和心血管疾病的疾病。 本发明还涉及可用于制备所述羧酸衍生物的中间体和制备方法。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D263/00 | 杂环化合物,含有1,3-唑环或氢化1,3-唑环 |
--------C07D263/02 | .不和其他环稠合 |
----------C07D263/04 | ..环原子间或环原子与非环原子间没有双键 |
------------C07D263/32 | ...只有氢原子、烃基或取代烃基,直接连在环碳原子上 |