发明申请
WO2004009073A1 P-GLYCOPROTEIN INHIBITOR COMPRISING OCTILONIUM BROMIDE AS AN EFFECTIVE INGREDIENT
审中-公开
基本信息:
- 专利标题: P-GLYCOPROTEIN INHIBITOR COMPRISING OCTILONIUM BROMIDE AS AN EFFECTIVE INGREDIENT
- 专利标题(中):含有作为有效成分的溴氰菊酯的P-糖蛋白抑制剂
- 申请号:PCT/KR2003/001441 申请日:2003-07-21
- 公开(公告)号:WO2004009073A1 公开(公告)日:2004-01-29
- 发明人: CHUNG, Hesson , JEONG, Seo-Young , KWON, Ick-Chan , PARK, Yeong-Taek , LEE, In-Hyun , YUK, Soon-Hong
- 申请人: KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY , CHUNG, Hesson , JEONG, Seo-Young , KWON, Ick-Chan , PARK, Yeong-Taek , LEE, In-Hyun , YUK, Soon-Hong
- 申请人地址: 39-1, Hawolgok-Dong, Sungbook-Gu, Seoul 136-791 KR
- 专利权人: KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY,CHUNG, Hesson,JEONG, Seo-Young,KWON, Ick-Chan,PARK, Yeong-Taek,LEE, In-Hyun,YUK, Soon-Hong
- 当前专利权人: KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY,CHUNG, Hesson,JEONG, Seo-Young,KWON, Ick-Chan,PARK, Yeong-Taek,LEE, In-Hyun,YUK, Soon-Hong
- 当前专利权人地址: 39-1, Hawolgok-Dong, Sungbook-Gu, Seoul 136-791 KR
- 代理机构: PARK, Jang-Won
- 优先权: KR10-2002-0042794 20020720
- 主分类号: A61K31/245
- IPC分类号: A61K31/245
摘要:
The present invention relates to a new use of octylonium bromide as p-glycoprotein inhibitor to increase cellular uptake of drugs. More particularly, the present invention provides octylonium bromide as a p-glycoprotein inhibitor to increase cellular uptake of drugs such as anticancer drugs by taking octylonium bromide simultaneously with or proceding drug administration.
摘要(中):
本发明涉及辛基溴化物作为P-糖蛋白抑制剂的新用途,以增加药物的细胞吸收。 更具体地,本发明提供了作为P-糖蛋白抑制剂的辛基溴化铵,以通过同时服用辛基溴或同时给予药物来增加药物如抗癌药物的细胞摄取。
IPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K31/00 | 含有机有效成分的医药配制品 |
--------A61K31/045 | .羟基化合物,例如醇类;其盐类,例如醇化物 |
----------A61K31/215 | ..羧酸酯 |
------------A61K31/22 | ...无环酸的酯,例如帕伐他丁 |
--------------A61K31/24 | ....有1个氨基或硝基的 |
----------------A61K31/245 | .....氨基苯甲酸型,例如普鲁卡因,奴夫卡因 |