基本信息:
- 专利标题: PYRROLE-2, 5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS
- 申请号:PCT/US2003/005052 申请日:2003-03-05
- 公开(公告)号:WO2003076398A3 公开(公告)日:2003-09-18
- 发明人: ALBAUGH, Pamela, Ann , AMMENN, Jochen , BURKHOLDER, Timothy, Paul , CLAYTON, Joshua, Ryan , CONNER, Scott, Eugene , CUNNINGHAM, Brian, Eugene , ENGLER, Thomas, Albert , FURNESS, Kelly, Wayne , HENRY, James, Robert , LI, YiHong , MALHOTRA, Sushant , TEBBE, Mark, Joseph , ZHU, Guoxin
- 申请人: ELI LILLY AND COMPANY , ALBAUGH, Pamela, Ann , AMMENN, Jochen , BURKHOLDER, Timothy, Paul , CLAYTON, Joshua, Ryan , CONNER, Scott, Eugene , CUNNINGHAM, Brian, Eugene , ENGLER, Thomas, Albert , FURNESS, Kelly, Wayne , HENRY, James, Robert , LI, YiHong , MALHOTRA, Sushant , TEBBE, Mark, Joseph , ZHU, Guoxin
- 申请人地址: Lilly Corporate Center, Indianapolis, IN 46285 US
- 专利权人: ELI LILLY AND COMPANY,ALBAUGH, Pamela, Ann,AMMENN, Jochen,BURKHOLDER, Timothy, Paul,CLAYTON, Joshua, Ryan,CONNER, Scott, Eugene,CUNNINGHAM, Brian, Eugene,ENGLER, Thomas, Albert,FURNESS, Kelly, Wayne,HENRY, James, Robert,LI, YiHong,MALHOTRA, Sushant,TEBBE, Mark, Joseph,ZHU, Guoxin
- 当前专利权人: ELI LILLY AND COMPANY,ALBAUGH, Pamela, Ann,AMMENN, Jochen,BURKHOLDER, Timothy, Paul,CLAYTON, Joshua, Ryan,CONNER, Scott, Eugene,CUNNINGHAM, Brian, Eugene,ENGLER, Thomas, Albert,FURNESS, Kelly, Wayne,HENRY, James, Robert,LI, YiHong,MALHOTRA, Sushant,TEBBE, Mark, Joseph,ZHU, Guoxin
- 当前专利权人地址: Lilly Corporate Center, Indianapolis, IN 46285 US
- 代理机构: TITUS, Robert, D.
- 优先权: US60/363,375 20020308; US60/369,433 20020402
- 主分类号: C07D401/14
- IPC分类号: C07D401/14
摘要:
The present invention provides kinase inhibitors of Formula (I)
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D401/00 | 杂环化合物,含有两个或更多个杂环,以氮原子作为仅有的杂环原子,至少有1个环是仅含有1个氮原子的六元环 |
--------C07D401/14 | .含有3个或更多个杂环 |