基本信息:
- 专利标题: HYDROXY ACID INTEGRIN ANTAGONISTS
- 申请号:PCT/US2001/030189 申请日:2001-09-27
- 公开(公告)号:WO2002026717A3 公开(公告)日:2002-04-04
- 发明人: ROGERS, Thomas , PENNING, Thomas, D. , LAN, Jiang , DEVADAS, Balekudru , RUMINISKI, Peter , YUAN, Chester , VANCAMP, Jennifer
- 申请人: PHARMACIA CORPORATION , ROGERS, Thomas , PENNING, Thomas, D. , LAN, Jiang , DEVADAS, Balekudru , RUMINISKI, Peter , YUAN, Chester , VANCAMP, Jennifer
- 申请人地址: 800 N. Lindbergh, Mail Zone O4E, St. Louis, MO 63167 US
- 专利权人: PHARMACIA CORPORATION,ROGERS, Thomas,PENNING, Thomas, D.,LAN, Jiang,DEVADAS, Balekudru,RUMINISKI, Peter,YUAN, Chester,VANCAMP, Jennifer
- 当前专利权人: PHARMACIA CORPORATION,ROGERS, Thomas,PENNING, Thomas, D.,LAN, Jiang,DEVADAS, Balekudru,RUMINISKI, Peter,YUAN, Chester,VANCAMP, Jennifer
- 当前专利权人地址: 800 N. Lindbergh, Mail Zone O4E, St. Louis, MO 63167 US
- 代理机构: POLSTER, Rachel, A.
- 优先权: US60/235,616 20000927; US60/241,656 20001019
- 主分类号: C07D239/14
- IPC分类号: C07D239/14
摘要:
The present invention relates to compounds, pharmaceutical compositions and method of using α v β 3 and/or α v β 5 selective integrin antagonists.
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D239/00 | 杂环化合物,含1,3-二嗪环或氢化1,3-二嗪环 |
--------C07D239/02 | .不与其他环稠合 |
----------C07D239/06 | ..环原子间或环原子与非环原子间有1个双键 |
------------C07D239/08 | ...有杂原子直接连在位置2 |
--------------C07D239/12 | ....非硝基氮原子 |
----------------C07D239/14 | .....只有氢原子、烃基或取代的烃基,连在上述氮原子上 |