发明申请
WO1995021833A1 SUBSTITUTED OXAZACYCLOALKENES, INTERMEDIATE PRODUCTS AND USE AS FUNGICIDES
审中-公开
基本信息:
- 专利标题: SUBSTITUTED OXAZACYCLOALKENES, INTERMEDIATE PRODUCTS AND USE AS FUNGICIDES
- 专利标题(中):取代OXAZACYCLOALKENE,中间体和使用作为杀真菌剂
- 申请号:PCT/EP1995000311 申请日:1995-01-30
- 公开(公告)号:WO1995021833A1 公开(公告)日:1995-08-17
- 发明人: BAYER AKTIENGESELLSCHAFT
- 申请人: BAYER AKTIENGESELLSCHAFT , SEITZ, Thomas , ASSMANN, Lutz , GAYER, Herbert , GERDES, Peter , HEINEMANN, Ulrich , KRÜGER, Bernd-Wieland , KUHNT, Dietmar , TIEMANN, Ralf , DEHNE, Heinz-Wilhelm , DUTZMANN, Stefan , HÄNSSLER, Gerd , STENZEL, Klaus
- 专利权人: BAYER AKTIENGESELLSCHAFT,SEITZ, Thomas,ASSMANN, Lutz,GAYER, Herbert,GERDES, Peter,HEINEMANN, Ulrich,KRÜGER, Bernd-Wieland,KUHNT, Dietmar,TIEMANN, Ralf,DEHNE, Heinz-Wilhelm,DUTZMANN, Stefan,HÄNSSLER, Gerd,STENZEL, Klaus
- 当前专利权人: BAYER AKTIENGESELLSCHAFT,SEITZ, Thomas,ASSMANN, Lutz,GAYER, Herbert,GERDES, Peter,HEINEMANN, Ulrich,KRÜGER, Bernd-Wieland,KUHNT, Dietmar,TIEMANN, Ralf,DEHNE, Heinz-Wilhelm,DUTZMANN, Stefan,HÄNSSLER, Gerd,STENZEL, Klaus
- 优先权: DEP 19940211
- 主分类号: C07D265/08
- IPC分类号: C07D265/08
摘要:
Substituted oxazacycloalkenes of formula (I) in which A is optionally substituted alkane diyl (alkylene), Ar is optionally substituted arylene or heteroarylene; E is a 1-alkene-1,1-diyl group containing a radical R in the 2nd position or a 2-aza-1-alkene-1,1-diyl group containing a radical R in the 2nd position, or a 3-aza-1-propene-2,3-diyl group containing a radical R in the 3rd position and a radical R in the 1st position, or a 1-aza-1-propene-2,3-diyl group containing a radical R in the 1st position, or a 1,3-diaza-1-propene-2,3-diyl group containing a radical R in the 3rd position and a radical R in the 1st position, or an optionally substituted imino group ("azamethylene", N-R ), G is oxygen or, optionally substituted by halogen, hydroxy, alkyl, halogen alkyl or cycloalkyl, alkane diyl or one of the groups: -Q-CQ-, -CQ-Q-, -CH2-Q-, -Q-CH2-, -CQ-Q-CH2-, -CH2-Q-CQ-, -Q-CQ-CH2-, -Q-CQ-Q-CH2-, -N=N-, -S(O)n-, -CH2-S(O)n-, -CQ-, -S(O)n-CH2-, -C(R )=N-O-, -C(R )=N-O-CH2-, -N(R )-, -CQ-N(R )-, -N(R )-CQ-, -Q-CQ-N(R )-, -N=C(R )-Q-CH2-, -CH2-O-N=C(R )-, -N(R )-CQ-Q-, -CQ-N(R )-CQ-Q-, -N(R )-CQ-Q-CH2-, -CQ-CH2- oder -N=N-C(R )=N-O-; Z is optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, aryl or heterocyclyl, a process for their production and the use of oxazacycloalkenes as fungicides.
摘要(中):
取代的式(I),其中A代表任选取代的烷二基(亚烷基),Ar是任选取代的亚芳基或亚杂芳基的Oxazacycloalkene,E表示的1-烯烃-1,1-二基分组这在2- 定位一个基团R <1>包含,或者是2-氮杂-1-链烯-1,1-二基分组其中基团R <2>包含2位或3-氮杂 其中基团R和1位在位置3包含一个基团R <1>,或代表1-氮杂-1-丙烯-2,3-二基部分的丙烯-2,3-二基分组 是一个基团R <2>包含在1-位,或表示1,3-二氮杂-1-丙烯-2,3-二基,其分组在3位的基团R和在1-位 一个基团R <2>包含,或(“azamethylene”,NR <3>)是任选取代的亚氨基,G表示氧,在每种情况下任选地被卤素,羟基,烷基,卤代烷基或环烷基取代的烷二基,或其中一个取代的 下面-Q-CQ-分组是,-CQ-Q-,-CH 2 -Q-,-Q-CH 2 - ,-CQ-Q-CH2-,-CH2-Q-CQ-,-Q-CQ-CH2- ,-Q-CQ-Q-CH 2 - , - N = N-,-S(O)N-,-CH 2 S(O)N-,-CQ-,-S(O)N-CH 2 - , - C(R <4>)= NO-,-C(R <4>)= NO-CH 2 - ,-N(R <5>) - ,-CQ-N(R <5>) - , - N( [R <5>) - CQ-,-Q-CQ-N(R <5>) - , - N = C(R <4>) - Q-CH2-,-CH2-ON = C(R <4> ) - , - N(R <5>) - CQ-Q-,-CQ-N(R <5>) - CQ-Q,-N(R <5>) - CQ-Q-CH2 - CQ-CH 2或-N = NC(R <4>)= NO-,Z代表任选取代的烷基,烯基,炔基,环烷基,芳基或杂环基,一种方法和用于制备它们的中间体和使用作为Oxazacycloalkenen 杀菌剂。
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D265/00 | 杂环化合物,含六元环,有1个氮原子和1个氧原子作为仅有的杂环原子 |
--------C07D265/04 | .1,3-嗪;氢化1,3-嗪 |
----------C07D265/06 | ..不与其他环稠合 |
------------C07D265/08 | ...环原子间或环原子与非环原子间有1个双键 |