发明申请
US20200172547A1 TRIAZOLO[4,5-D] PYRAMIDINE DERIVATIVES AND THEIR USE AS PURINE RECEPTOR ANTAGONISTS
审中-公开
![TRIAZOLO[4,5-D] PYRAMIDINE DERIVATIVES AND THEIR USE AS PURINE RECEPTOR ANTAGONISTS](/abs-image/US/2020/06/04/US20200172547A1/abs.jpg.150x150.jpg)
基本信息:
- 专利标题: TRIAZOLO[4,5-D] PYRAMIDINE DERIVATIVES AND THEIR USE AS PURINE RECEPTOR ANTAGONISTS
- 申请号:US16700160 申请日:2019-12-02
- 公开(公告)号:US20200172547A1 公开(公告)日:2020-06-04
- 发明人: Samantha Jane Bamford , Roger John Gillespie , Richard Simon Todd
- 申请人: Vernalis (R&D) Limited
- 申请人地址: GB Winnersh
- 专利权人: Vernalis (R&D) Limited
- 当前专利权人: Vernalis (R&D) Limited
- 当前专利权人地址: GB Winnersh
- 优先权: com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@10c22ae8
- 主分类号: C07D487/04
- IPC分类号: C07D487/04 ; A61K31/197 ; A61K31/519 ; A61K45/06 ; C07D405/12
摘要:
Compounds of formula (I) that are capable of acting as purine receptor antagonists, pharmaceutical compositions including the compounds, and methods of making the compounds, are. disclosed. The compounds and compositions can be used in treating or preventing disorders related to purine receptor hyperfunctioning.
公开/授权文献:
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D487/00 | 在稠环系中含有氮原子作为仅有的杂环原子的杂环化合物,不包含在C07D451/00至C07D477/00组中 |
--------C07D487/02 | .在稠合系中含有两个杂环 |
----------C07D487/04 | ..邻位稠合系 |