基本信息:
- 专利标题: 좌심실 확장 기능 개선제
- 专利标题(英):Left ventricular diastolic function improving agent
- 专利标题(中):左心室肌纤维功能改善剂
- 申请号:KR1020147002583 申请日:2012-08-01
- 公开(公告)号:KR1020140056250A 公开(公告)日:2014-05-09
- 发明人: 가나지도시야 , 후치베가즈히로 , 다카하시마사야
- 申请人: 오노 야꾸힝 고교 가부시키가이샤
- 申请人地址: 일본국오사카후오사카시츄오쿠도쇼마치* 쪼메*반*고
- 专利权人: 오노 야꾸힝 고교 가부시키가이샤
- 当前专利权人: 오노 야꾸힝 고교 가부시키가이샤
- 当前专利权人地址: 일본국오사카후오사카시츄오쿠도쇼마치* 쪼메*반*고
- 代理人: 김진회
- 优先权: JPJP-P-2011-169389 2011-08-02
- 国际申请: PCT/JP2012/069609 2012-08-01
- 国际公布: WO2013018837 2013-02-07
- 主分类号: A61K31/4015
- IPC分类号: A61K31/4015 ; A61K47/40 ; A61K38/22 ; A61P1/16
The present invention, heart failure, a therapeutic agent that can be irrespective of the diuretic and vasodilating action to improve the extension of the left ventricle itself, prevent the recurrence by controlling the conditions of the expansion insufficiency, improving the dyspnea and mortality according to the same conditions to provide an object. 4 - [(2 - {(2R) -2 - [(1E, 3S) -4- (4-fluorophenyl) -3-hydroxy-1-buten-1-yl] -5-oxo-1 pyrrolidinyl} ethyl) thio] butane acid, by directly acting on the heart, among improve extension of the left ventricle and heart failure, in particular, can be effectively treated to expand insufficiency. Thus, it is possible to provide a new heart failure therapeutic agent that can by the present invention, to improve the expansion dysfunction not established a valid treatment.
信息查询:
EspacenetIPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K31/00 | 含有机有效成分的医药配制品 |
--------A61K31/33 | .杂环化合物 |
----------A61K31/335 | ..仅有氧作为环杂原子的,例如制霉色基素 |
------------A61K31/40 | ...有仅以1个氮作为环杂原子的五元环的,例如舒必利、琥珀酰亚胺、托尔米丁、甲氧吡丁苯 |
--------------A61K31/4015 | ....含有直接与杂环相连的氧代基团的,例如脑复康、乙琥胺 |