基本信息:
- 专利标题: 항미생물성 아미노-살리실산 유도체
- 专利标题(英):Antimicrobial amino-salicylic acid derivatives
- 申请号:KR1020127007512 申请日:2010-08-13
- 公开(公告)号:KR101759360B1 公开(公告)日:2017-07-18
- 发明人: 홀즐,베르너 , 푸르츠비츠,야니나
- 申请人: 바스프 에스이
- 申请人地址: Carl-Bosch-Strasse **, ***** Ludwigshafen am Rhein, Germany
- 专利权人: 바스프 에스이
- 当前专利权人: 바스프 에스이
- 当前专利权人地址: Carl-Bosch-Strasse **, ***** Ludwigshafen am Rhein, Germany
- 代理人: 양영준; 위혜숙
- 优先权: EP091686691 2009-08-26
- 国际申请: PCT/EP2010/061804 2010-08-13
- 国际公布: WO2011023573 2011-03-03
- 主分类号: A61K31/167
- IPC分类号: A61K31/167 ; A61K8/42 ; A61K8/44 ; C11D3/48 ; C11D3/32 ; A61Q17/00 ; A61Q5/02 ; A61Q11/02 ; A61Q15/00
This new way of achieving the object and / or protection in the substance or object and / or anti-microbial effect for the protection of material on the surface, preserving effect, and / or microbial adhesion inhibitory effect is described. The present new method comprises applying a salicylic acid compound, or a salt or adduct of the formula (I) to the object and / or substance.
<Formula I>
Wherein
A and A 'is one of the formula I' is the residue of,
-NH-CO-R 1 (I ')
The other is hydrogen;
R
1 is C
1 -C
22 alkyl, C
3 -C
12 cycloalkyl, O and / or NR
5 is interposed a C
3 -C
12 cycloalkyl, C
4 -C
12 aryl, C
5 -C
18 aryl and .;
R
2 is OR
3 or NHR
4, and;
R
3 and R
4 are H, C
1 -C
22 alkyl, C
3 -C
12 cycloalkyl, O and / or NR
5 is interposed a C
3 -C
12 cycloalkyl, C
4 -C
12 aryl, C
5 - C
18 aryl alkyl;
R
5 is H or C
1 -C
8 alkyl;
Wherein each aryl moiety is unsubstituted or substituted by C
1 -C
4 alkyl, C
1 -C
4 alkoxy, C
1 -C
4 acyl, C
1 -C
4 acyloxy, C
1 -C
4 acylamino, CF
3 and it is optionally substituted by OH, amino, halogen.
公开/授权文献:
- KR1020120055712A 항미생물성 아미노-살리실산 유도체 公开/授权日:2012-05-31
信息查询:
EspacenetIPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K31/00 | 含有机有效成分的医药配制品 |
--------A61K31/045 | .羟基化合物,例如醇类;其盐类,例如醇化物 |
----------A61K31/165 | ..含芳环的,例如秋水仙碱、阿替洛尔、氟柳双胺 |
------------A61K31/167 | ...甲酰胺的氮原子直接与芳环相连的,例如利多卡因、对乙酰氨基酚 |