基本信息:
- 专利标题： IMIDAZOPYRIMIDINE DERIVATIVE AND TRIAZOLOPYRIMIDINE DERIVATIVE
- 申请号：JP2000128870 申请日：2000-04-28
- 公开(公告)号：JP2001302667A 公开(公告)日：2001-10-31
- 发明人： YURA TAKESHI , ARNEL B CONCEPTION , KAN KINKI , HIRAOKA MAKIKO , KATSUMATA HIROKO , KAWAMURA NORIHIRO , KOKUBO TOSHIO , KOMURA HIROSHI , RI EIFU , TIMOTHY B ROOWINJAA , MOGI MUNEHITO , YAMAMOTO TOMOYUKI , YOSHIDA NAGAHIRO
- 申请人： BAYER AG
- 专利权人： BAYER AG
- 当前专利权人： BAYER AG
- 优先权： JP2000128870 2000-04-28
- 主分类号： A61K31/505
- IPC分类号： A61K31/505 ; A61K31/519 ; A61K31/5377 ; A61K31/541 ; A61P1/04 ; A61P3/04 ; A61P7/02 ; A61P7/06 ; A61P11/02 ; A61P11/06 ; A61P17/00 ; A61P17/04 ; A61P17/06 ; A61P19/02 ; A61P21/04 ; A61P25/28 ; A61P27/02 ; A61P27/14 ; A61P29/00 ; A61P35/00 ; A61P37/02 ; A61P37/06 ; A61P37/08 ; A61P43/00 ; C07D487/04 ; C07D519/00
摘要：
PROBLEM TO BE SOLVED: To provide a compound exhibiting excellent Syk tyrosine kinase inhibiting activity. SOLUTION: The objective compound is expressed by formula (R1 is X-R4, a (substituted) heterocyclic group, a (substituted) carbocyclic group or a (substituted) condensed ring group; X is CR5R6, O, S, SO, SO2 or NR7, Y is CH or N; R2 is H, a (substituted) 1-10C alkyl or the like; R3 is a (substituted) aryl, a (substituted) heteroaryl or the like; R4 is a (substituted) aryl, a (substituted) heteroaryl or the like; and R5, R6 and R7 are each independently H, a (substituted) 1-10C alkyl or the like).
信息查询:
EspacenetIPC结构图谱:
| A | 人类生活必需 |
| --A61 | 医学或兽医学；卫生学 |
| ----A61K | 医用、牙科用或梳妆用的配制品 |
| ------A61K31/00 | 含有机有效成分的医药配制品 |
| --------A61K31/33 | .杂环化合物 |
| ----------A61K31/335 | ..仅有氧作为环杂原子的，例如制霉色基素 |
| ------------A61K31/40 | ...有仅以1个氮作为环杂原子的五元环的，例如舒必利、琥珀酰亚胺、托尔米丁、甲氧吡丁苯 |
| --------------A61K31/505 | ....嘧啶；氢化嘧啶，例如甲氧苄啶 |