发明公开
EP3066106A1 STABLE PANTETHEINE DERIVATIVES FOR THE TREATMENT OF PANTOTHENATE KINASE ASSOCIATED NEURODEGENERATION (PKAN) AND METHODS FOR THE SYNTHESIS OF SUCH COMPOUNDS
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基本信息:
- 专利标题: STABLE PANTETHEINE DERIVATIVES FOR THE TREATMENT OF PANTOTHENATE KINASE ASSOCIATED NEURODEGENERATION (PKAN) AND METHODS FOR THE SYNTHESIS OF SUCH COMPOUNDS
- 专利标题(中):稳定PANTETHEINDERIVATE与泛酸激酶相关性神经变性(PKAN)和方法请客合成等环节
- 申请号:EP14790616.8 申请日:2014-10-29
- 公开(公告)号:EP3066106A1 公开(公告)日:2016-09-14
- 发明人: JENKO, Branko , KOSEC, Gregor , PETKOVIC, Hrvoje , PODGORSEK BERKE, Ajda , PAHOR, Jerca , CUSAK, Alen , SIBON, Oda Cornelia Maria , SRINIVASAN, Balaji
- 申请人: Acies Bio d.o.o. , Rijksuniversiteit te Groningen , Academisch Ziekenhuis Groningen
- 申请人地址: Tehnoloski park 21 1000 Ljubljana SI
- 专利权人: Acies Bio d.o.o.,Rijksuniversiteit te Groningen,Academisch Ziekenhuis Groningen
- 当前专利权人: VECTIVBIO COMET AG, CH
- 当前专利权人地址: VECTIVBIO COMET AG, CH
- 代理机构: Zacco GmbH
- 优先权: EP13191457 20131104
- 国际公布: WO2015063177 20150507
- 主分类号: C07F9/09
- IPC分类号: C07F9/09 ; A61K31/661 ; A61P25/28
摘要:
The invention relates to (S)-acyl-4'-phosphopantetheine derivatives, methods of their synthesis, and related medical uses of such compounds. Preferred medical uses relate to the treatment ofneurodegenerative diseases, such as PKAN.
摘要(中):
本发明涉及(S)酰基-4'-磷酸泛酰衍生物,它们的合成的方法,以及测试化合物相关的医疗用途。 优选的医疗用途涉及治疗疾病ofneurodegenerative ,:如PKAN。