发明公开
EP2552909A1 4 - AMINOPYRIMIDINE DERIVATIVES AND THEIR AS AS ADENOSINE A2A RECEPTOR ANTAGONISTS
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基本信息:
- 专利标题： 4 - AMINOPYRIMIDINE DERIVATIVES AND THEIR AS AS ADENOSINE A2A RECEPTOR ANTAGONISTS
- 专利标题（中）：4 - 氨基嘧啶衍生物及其作为腺苷A2A受体拮抗剂使用
- 申请号：EP11719879.6 申请日：2011-03-29
- 公开(公告)号：EP2552909A1 公开(公告)日：2013-02-06
- 发明人： CAMACHO GOMEZ, Juan Alberto , CASTRO-PALOMINO LARIA, Julio Cesar
- 申请人： Palobiofarma, S.L.
- 申请人地址： C/Porvenir 42 Pol.Ind.Sur, Sector F 08450 Llinars del Vallès ES
- 专利权人： Palobiofarma, S.L.
- 当前专利权人： PALOBIOFARMA S.L.
- 当前专利权人地址： PALOBIOFARMA S.L.
- 代理机构： Maldonado Jordan, Julia
- 优先权： ES201030489 20100331
- 国际公布： WO2011121418 20111006
- 主分类号： C07D403/04
- IPC分类号： C07D403/04 ; C07D403/14 ; C07D409/14 ; C07D413/14 ; C07D417/04 ; C07D417/14 ; A61K31/506 ; A61P3/10 ; A61P25/00
摘要：
New 4-amino-pyrimidine derivatives as potent antagonists of the adenosine A
2a receptor formula (I): (I) The invention provides as well a method for preparing such compounds, pharmaceutical compositions comprising an effective amount of these compounds and the use of such compounds in the manufacture of a medicament to treat pathological affections that can be improved by antagonism of the adenosine A
2a receptor.
2a receptor formula (I): (I) The invention provides as well a method for preparing such compounds, pharmaceutical compositions comprising an effective amount of these compounds and the use of such compounds in the manufacture of a medicament to treat pathological affections that can be improved by antagonism of the adenosine A
2a receptor.
公开/授权文献:
IPC结构图谱:
| C | 化学；冶金 |
| --C07 | 有机化学 |
| ----C07D | 杂环化合物 |
| ------C07D403/00 | 杂环化合物，含有两个或更多的杂环，以氮原子作为仅有的杂环原子，C07D401/00组不包含的 |
| --------C07D403/02 | .含两个杂环 |
| ----------C07D403/04 | ..被环原子—环原子的键直接连接的 |