发明公开
EP0045118A3 Intermediates for the synthesis of bicyclo (2,2,1) heptanes and bicyclo (2,2,1) hept-2Z-enes
有权
转让
基本信息:
- 专利标题： Intermediates for the synthesis of bicyclo (2,2,1) heptanes and bicyclo (2,2,1) hept-2Z-enes
- 专利标题（中）：二氨基（2,2,1）庚二酸和二巯基（2,2,1）HEPT-2Z-烯的合成中间体
- 申请号：EP81201031 申请日：1980-01-04
- 公开(公告)号：EP0045118A3 公开(公告)日：1982-03-24
- 发明人： Jones, Robert Leslie
- 申请人： Jones, Robert Leslie , Wilson, Norman Happer
- 专利权人： Jones, Robert Leslie,Wilson, Norman Happer
- 当前专利权人： BRITISH TECHNOLOGY GROUP LTD TE LONDEN, GROOT-BRIT
- 当前专利权人地址： BRITISH TECHNOLOGY GROUP LTD TE LONDEN, GROOT-BRIT
- 优先权： GB7900368 19790105
- 主分类号： C07C59/11
- IPC分类号： C07C59/11 ; C07C59/205 ; C07C59/46 ; C07C59/80 ; C07C177/00
摘要：
Novel bicyclo[2,2,1]heptanes and hept-2Z-enes are substituted at the 5-position by a 6-carboxyhex-2-enyl group or a modification thereof as defined herein, and at the 6-position by a group
in which R 1 represents an aliphatic hydrocarbon residue or an aliphatic hydrocarbon residue substituted directly or through an oxygen or sulphur atom by an aromatic residue, R2 represents hydrogen and R 3 represents a hydroxy group, or R 2 and R 3 together represent the oxygen atom of a carboxyl group. These compounds are of value for use in the synthesis of certain biologically active 5,6-disubstituted bicyclo[2,2,1]heptanes and hept-2Z-enes.
摘要（中）：
in which R 1 represents an aliphatic hydrocarbon residue or an aliphatic hydrocarbon residue substituted directly or through an oxygen or sulphur atom by an aromatic residue, R2 represents hydrogen and R 3 represents a hydroxy group, or R 2 and R 3 together represent the oxygen atom of a carboxyl group. These compounds are of value for use in the synthesis of certain biologically active 5,6-disubstituted bicyclo[2,2,1]heptanes and hept-2Z-enes.
新的双环[2,2,1]庚烷和庚-2Z-烯通过如本文所定义的6-羧基己-2-烯基或其修饰在5位上被取代，并且在6-位上被一个基团 其中R1表示脂肪族烃残基或由芳香族残基直接或通过氧或硫原子取代的脂族烃残基，R2表示氢，R3表示羟基，或R2和R3一起代表 羧基。 这些化合物对于合成某些生物活性的5,6-二取代的双环[2,2,1]庚烷和庚-2Z-烯有价值。