发明专利
CA2836316A1 HYDROXYLATED AND METHOXYLATED CYCLOPENTA [D] PYRIMIDINES AS AKT PROTEIN KINASE INHIBITORS
未知
基本信息:
- 专利标题: HYDROXYLATED AND METHOXYLATED CYCLOPENTA [D] PYRIMIDINES AS AKT PROTEIN KINASE INHIBITORS
- 申请号:CA2836316 申请日:2007-07-05
- 公开(公告)号:CA2836316A1 公开(公告)日:2008-01-10
- 发明人: MITCHELL IAN S , BLAKE JAMES F , XU RUI , KALLAN NICHOLAS C , XIAO DENGMING , SPENCER KEITH LEE , BENCSIK JOSEF R , LIANG JUN , SAFINA BRIAN , ZHANG BIRONG , CHABOT CHRISTINE , DO STEVEN , WALLACE ELI M , BANKA ANNA L , SCHLACHTER STEPHEN T
- 申请人: ARRAY BIOPHARMA INC , GENENTECH INC
- 专利权人: ARRAY BIOPHARMA INC,GENENTECH INC
- 当前专利权人: ARRAY BIOPHARMA INC,GENENTECH INC
- 优先权: US81871806 2006-07-06
- 主分类号: C07D403/02
- IPC分类号: C07D403/02 ; A61K31/517 ; C07C229/34
摘要:
The present invention provides compounds, including resolved enantiomers, resolved diastereomers, solvates and pharmaceutically acceptable salts thereof, comprising the Formula (I). Also provided are methods of using the compounds of this invention as AKT protein kinase inhibitors and for the treatment of hyperproliferative diseases such as cancer. (see formula I)
信息查询:
EspacenetIPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D403/00 | 杂环化合物,含有两个或更多的杂环,以氮原子作为仅有的杂环原子,C07D401/00组不包含的 |
--------C07D403/02 | .含两个杂环 |