基本信息:
- 专利标题: Bis 2'-5'-RR-(3'F-A)(3'F-A) cyclic dinucleotide compound and uses thereof
- 申请号:AU2018260494 申请日:2018-04-26
- 公开(公告)号:AU2018260494A1 公开(公告)日:2019-11-07
- 发明人: LEONG JUSTIN , NDUBAKU CHUDI OBIOMA , MCKENNA JEFFREY
- 申请人: ADURO BIOTECH INC , NOVARTIS AG
- 专利权人: ADURO BIOTECH INC,NOVARTIS AG
- 当前专利权人: ADURO BIOTECH INC,NOVARTIS AG
- 优先权: US201762578172 2017-10-27; US201762491879 2017-04-28
- 主分类号: C07H21/02
- IPC分类号: C07H21/02 ; A61K31/7084 ; A61K47/26 ; A61P35/00
摘要:
The present invention provides the cyclic dinucleotide compound 2'2'-RR-(3'F-A)(3'F- A) as a highly active immune stimulator that activates DCs via the cytoplasmic receptor known as STING (Stimulator of Interferon Genes), and compositions and uses thereof.
信息查询:
EspacenetIPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07H | 糖类;及其衍生物;核苷;核苷酸;核酸 |
------C07H21/00 | 含有两个或多个单核苷酸单元的化合物,具有以核苷基的糖化物基团连接的单独的磷酸酯基或多磷酸酯基,例如核酸 |
--------C07H21/02 | .以核糖基作为糖化物基团 |